SCHEMBL2169907

SCHEMBL2169907

COc1ccc(Oc2c(Cl)cc(C=O)cc2Cl)cc1C(C)C

nearest known ligand 0.65

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
RORC P51449 10/20 0.65
THRB P10828 10/20 0.65
THRA P10827 5/20 0.47
HTT P42858 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16495807 0.88 THRB (0.54) RORCTHRBTHRAHTT
SCHEMBL282394 0.85 THRB (0.50) RORCTHRBTHRAHTT
SCHEMBL16496567 0.84 THRB (0.53) RORCTHRBTHRAHTT
SCHEMBL2169380 0.84 RORC (0.65) RORCTHRBTHRAHTT
SCHEMBL2169378 0.84 RORC (0.65) RORCTHRBTHRAHTT
SCHEMBL6818059 0.82 RORC (0.70) RORCTHRBTHRA
SCHEMBL22959261 0.82 THRB (0.70) RORCTHRBTHRA
SCHEMBL5619231 0.81 THRB (0.73) RORCTHRBTHRA
SCHEMBL281885 0.80 THRB (0.79) RORCTHRBTHRA
SCHEMBL22959356 0.80 RORC (0.67) RORCTHRBTHRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110301200-A1 THYROID RECEPTOR LIGANDS CADILA HEALTHCARE LIMITED (IN) 2011-12-08 US disclosed
EP-2346814-A2 THYROID RECEPTOR LIGANDS Cadila Healthcare Limited (IN) 2011-07-27 EP disclosed
WO-2010049946-A2 THYROID RECEPTOR LIGANDS CADILA HEALTHCARE LIMITED (IN) 2010-05-06 WO disclosed
EP-1148054-B1 Thyroid receptor ligands PFIZER PROD INC (US) 2005-11-23 EP disclosed
US-6960604-B2 Thyroid receptor ligands PFIZER INC. (US) 2005-11-01 US disclosed
US-20040110951-A1 Thyroid receptor ligands CHIANG YUAN-CHING P (US) 2004-06-10 US disclosed
US-6620830-B2 Certain thiazolidinedione, oxadiazolidinedione, and triazolone compounds which are thyroid receptor ligands PFIZER, INC. 2003-09-16 US disclosed
US-20010051645-A1 Thyroid receptor ligands CHIANG YUAN-CHING P (US) 2001-12-13 US disclosed
EP-1148054-A1 Thyroid receptor ligands Pfizer Products Inc. (US) 2001-10-24 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110301200-A1 THYROID RECEPTOR LIGANDS TSHR, THRB, THRA RORC 79/4885THRB 2/4885THRA 3/4885
US-20010051645-A1 Thyroid receptor ligands TSHR, THRB, THRA RORC 302/4885THRB 2/4885THRA 3/4885
US-20040110951-A1 Thyroid receptor ligands TSHR, THRB, THRA RORC 302/4885THRB 2/4885THRA 3/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.