SCHEMBL21701238

SCHEMBL21701238

N#Cc1ccc(C(=O)N(CC2CC2)c2cccc(C(=O)Nc3c(I)cc(C(F)(C(F)(F)F)C(F)(F)F)cc3C(F)(F)F)c2F)cc1

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
RXFP1 Q9HBX9 2/20 0.37
HSD11B1 P28845 6/20 0.33
SMO Q99835 1/20 0.33
MLYCD O95822 1/20 0.33
HDAC8 Q9BY41 1/20 0.32
SLC6A2 P23975 1/20 0.32
SLC6A4 P31645 1/20 0.32
NSD2 O96028 2/20 0.32
MCHR1 Q99705 2/20 0.32
VNN1 O95497 1/20 0.32
KLKB1 P03952 1/20 0.31
GPBAR1 Q8TDU6 1/20 0.31
PDK2 Q15119 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22029433 0.92 HDAC8 (0.34) HSD11B1HDAC8SLC6A2SLC6A4GPBAR1
SCHEMBL21693605 0.91 RXFP1 (0.35) RXFP1HSD11B1SMOMLYCDHDAC8
SCHEMBL22029464 0.90 HDAC8 (0.35) RXFP1HSD11B1HDAC8SLC6A2SLC6A4
SCHEMBL23053028 0.90 FAAH (0.33) HDAC8GPBAR1
SCHEMBL23288057 0.89 RXFP1 (0.42) RXFP1HSD11B1SMOMLYCDHDAC8
SCHEMBL29857077 0.89 RXFP1 (0.42) RXFP1HSD11B1SMOMLYCDHDAC8
SCHEMBL24914654 0.88 RXFP1 (0.38) RXFP1MLYCDHDAC8VNN1
SCHEMBL24914954 0.88 RXFP1 (0.37) RXFP1MLYCDVNN1
SCHEMBL24626045 0.87 GPBAR1 (0.34) MLYCDHDAC8SLC6A2SLC6A4GPBAR1
SCHEMBL23053046 0.86 P2RX7 (0.37) MLYCDHDAC8GPBAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020030092-A1 PHARMACEUTICAL COMPOSITION CONTAINING M-DIAMIDE COMPOUND AND APPLICATION THEREOF 上海泰禾国际贸易有限公司 2020-02-13 WO disclosed
WO-2020030093-A1 PHARMACEUTICAL COMPOSITION CONTAINING M-DIAMIDE COMPOUND AND APPLICATION THEREOF 上海泰禾国际贸易有限公司 2020-02-13 WO disclosed