SCHEMBL2170428

SCHEMBL2170428

CC(NC(=O)CN1CCSC1)C(=O)Nc1ccc(Oc2ccc(F)cc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.47
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45
HPGD P15428 3/20 0.45
KDM4E B2RXH2 1/20 0.43
THRB P10828 1/20 0.43
ALOX15 P16050 1/20 0.42
S1PR1 P21453 1/20 0.42
LMNA P02545 1/20 0.42
GAA P10253 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
CHRNB2 P17787 2/20 0.41
CHRNB4 P30926 2/20 0.41
CHRNA3 P32297 2/20 0.41
CHRNA4 P43681 2/20 0.41
ATM Q13315 1/20 0.41
MAPT P10636 1/20 0.41
RECQL P46063 1/20 0.41
GLA P06280 1/20 0.40
REV1 Q9UBZ9 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2169800 0.94 ALDH1A1 (0.51) ALDH1A1MEN1KMT2AHPGDKDM4E
SCHEMBL2171842 0.84 ALDH1A1 (0.64) ALDH1A1MEN1KMT2AHPGDKDM4E
SCHEMBL2171615 0.84 ALDH1A1 (0.51) ALDH1A1MEN1KMT2AHPGDKDM4E
SCHEMBL2170390 0.83 SMN1; SMN2 (0.56) ALDH1A1MEN1KMT2AHPGDKDM4E
SCHEMBL2172990 0.82 ALDH1A1 (0.49) ALDH1A1MEN1KMT2AHPGDS1PR1
SCHEMBL1375590 0.80 S1PR1 (0.59) ALDH1A1MEN1KMT2AHPGDS1PR1
SCHEMBL1375592 0.80 S1PR1 (0.59) ALDH1A1MEN1KMT2AHPGDS1PR1
SCHEMBL2173707 0.80 MEN1 (0.50) ALDH1A1MEN1KMT2AHPGDKDM4E
SCHEMBL2185321 0.80 IDO1 (0.47) ALDH1A1MEN1KMT2AHPGDKDM4E
SCHEMBL2170253 0.77 ALDH1A1 (0.67) ALDH1A1MEN1KMT2AKDM4ETHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2349252-A2 SYNERGISTIC COMBINATION OF SPHINGOSINE-1-PHOSPHATE RECEPTOR ANTAGONISTS AND ANTIMICROTUBULE AGENTS Exelixis, Inc. (US) 2011-08-03 EP disclosed
EP-2346821-A1 SPHINGOSINE-1-PHOSPHATE RECEPTOR ANTAGONISTS Exelixis, Inc. (US) 2011-07-27 EP disclosed