SCHEMBL2170390

SCHEMBL2170390

CC1CCN(CC(=O)NC(C)C(=O)Nc2ccc(Oc3ccc(F)cc3)cc2)CC1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 5/20 0.56
ALDH1A1 P00352 9/20 0.50
MEN1 O00255 3/20 0.48
KMT2A Q03164 3/20 0.48
HPGD P15428 2/20 0.48
LMNA P02545 2/20 0.47
HTT P42858 1/20 0.47
KDM4E B2RXH2 3/20 0.47
TDP1 Q9NUW8 1/20 0.47
THRB P10828 1/20 0.46
ALOX15 P16050 1/20 0.46
MAPT P10636 2/20 0.45
GAA P10253 2/20 0.45
S1PR1 P21453 1/20 0.45
MAPK1 P28482 1/20 0.44
RAD52 P43351 1/20 0.44
GFER P55789 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
CHRNB2 P17787 2/20 0.44
CHRNB4 P30926 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2173707 0.88 MEN1 (0.50) SMN1; SMN2ALDH1A1MEN1KMT2AHPGD
SCHEMBL2171842 0.87 ALDH1A1 (0.64) ALDH1A1MEN1KMT2AHPGDKDM4E
SCHEMBL2169800 0.87 ALDH1A1 (0.51) SMN1; SMN2ALDH1A1MEN1KMT2AHPGD
SCHEMBL2171615 0.87 ALDH1A1 (0.51) SMN1; SMN2ALDH1A1MEN1KMT2AHPGD
SCHEMBL2185321 0.86 IDO1 (0.47) SMN1; SMN2ALDH1A1MEN1KMT2AHPGD
SCHEMBL2170428 0.83 ALDH1A1 (0.47) SMN1; SMN2ALDH1A1MEN1KMT2AHPGD
SCHEMBL3132407 0.82 ALDH1A1 (0.46) SMN1; SMN2ALDH1A1MEN1KMT2AHPGD
SCHEMBL2172990 0.82 ALDH1A1 (0.49) SMN1; SMN2ALDH1A1MEN1KMT2AHPGD
SCHEMBL2170963 0.81 MEN1 (0.48) ALDH1A1MEN1KMT2AHPGDLMNA
SCHEMBL1371825 0.81 S1PR1 (0.62) SMN1; SMN2ALDH1A1LMNAHTTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346821-A1 SPHINGOSINE-1-PHOSPHATE RECEPTOR ANTAGONISTS Exelixis, Inc. (US) 2011-07-27 EP disclosed