SCHEMBL21708751

SCHEMBL21708751

CCCC(F)OC(=O)CC(C#N)c1c(Cl)cccc1Cl

nearest known ligand 0.34

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.33
TAS1R3 Q7RTX0 1/20 0.32
TAS1R1 Q7RTX1 1/20 0.32
MEN1 O00255 3/20 0.32
ALDH1A1 P00352 2/20 0.32
LMNA P02545 2/20 0.32
HTT P42858 2/20 0.32
MAPT P10636 1/20 0.32
PKM P14618 1/20 0.32
NPSR1 Q6W5P4 1/20 0.31
HSD17B10 Q99714 1/20 0.31
RIPK1 Q13546 1/20 0.30
USP9X Q93008 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21708449 0.93 RIPK1 (0.36) KMT2AMEN1ALDH1A1LMNARIPK1
SCHEMBL21708518 0.89 TAS1R3 (0.32) KMT2ATAS1R3TAS1R1MEN1HSD17B10
SCHEMBL21708675 0.87 CCR1 (0.37) KMT2ATAS1R3TAS1R1MEN1ALDH1A1
SCHEMBL21708723 0.83 RIPK1 (0.36) KMT2AMEN1ALDH1A1LMNARIPK1
SCHEMBL21708777 0.82 KMT2A (0.38) KMT2AMEN1ALDH1A1MAPTNPSR1
SCHEMBL21708781 0.81 KMT2A (0.39) KMT2ATAS1R3TAS1R1HTTNPSR1
SCHEMBL21708792 0.79 TAS1R3 (0.33) KMT2ATAS1R3TAS1R1MEN1LMNA
SCHEMBL21708755 0.79 KMT2A (0.38) KMT2ATAS1R3TAS1R1MEN1ALDH1A1
SCHEMBL21708626 0.79 L3MBTL1 (0.30)
SCHEMBL21708728 0.78 KMT2A (0.39) KMT2AALDH1A1LMNAHTTMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3609869-A1 SUBSTITUTED N-ARYLETHYL-2-ARYLQUINOLINE-4-CARBOXAMIDES AND USE THEREOF Bayer Aktiengesellschaft (DE) 2020-02-19 EP disclosed