SCHEMBL21708792

SCHEMBL21708792

CCCC(F)OC(=O)CC(CN)c1c(Cl)cccc1Cl

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 1/20 0.33
TAS1R1 Q7RTX1 1/20 0.33
MEN1 O00255 4/20 0.32
KMT2A Q03164 4/20 0.32
GABBR2 O75899 4/20 0.31
GABBR1 Q9UBS5 4/20 0.31
LMNA P02545 2/20 0.31
CYP2C9 P11712 2/20 0.31
CYP3A4 P08684 1/20 0.31
ADORA3 P0DMS8 1/20 0.31
NFKB1 P19838 1/20 0.31
DRD3 P35462 1/20 0.31
BLM P54132 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C19 P33261 1/20 0.31
THRB P10828 1/20 0.31
TSHR P16473 1/20 0.31
HSD17B10 Q99714 1/20 0.31
NLRP3 Q96P20 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21708602 0.93 SMN1; SMN2 (0.33) MEN1KMT2ATSHR
SCHEMBL21708612 0.89 TAS1R3 (0.32) TAS1R3TAS1R1MEN1KMT2AHSD17B10
SCHEMBL21708646 0.86 NISCH (0.37) TAS1R3TAS1R1MEN1KMT2AGABBR2
SCHEMBL21708770 0.82 PTGFR (0.35) MEN1KMT2ALMNA
SCHEMBL21708787 0.82 HPGD (0.39) MEN1KMT2AGABBR2GABBR1LMNA
SCHEMBL21708747 0.80 TAS1R3 (0.36) TAS1R3TAS1R1KMT2ATSHR
SCHEMBL21708751 0.79 KMT2A (0.33) TAS1R3TAS1R1MEN1KMT2ALMNA
SCHEMBL21708683 0.78 F10 (0.38) TAS1R3TAS1R1GABBR2GABBR1CYP2C9
SCHEMBL21708509 0.78 NISCH (0.36) TAS1R3TAS1R1MEN1KMT2A
SCHEMBL21708638 0.77 GABBR2 (0.38) MEN1KMT2AGABBR2GABBR1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3609869-A1 SUBSTITUTED N-ARYLETHYL-2-ARYLQUINOLINE-4-CARBOXAMIDES AND USE THEREOF Bayer Aktiengesellschaft (DE) 2020-02-19 EP disclosed