SCHEMBL21708762

SCHEMBL21708762

CCCC(F)OC(=O)C(C)(C#N)c1ccccc1OC

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.37
MEN1 O00255 1/20 0.37
TSHR P16473 3/20 0.36
ATM Q13315 1/20 0.36
TAS1R3 Q7RTX0 1/20 0.34
TAS1R1 Q7RTX1 1/20 0.34
CTSS P25774 1/20 0.34
CTSK P43235 1/20 0.34
DPP4 P27487 1/20 0.33
FAP Q12884 1/20 0.33
GAA P10253 2/20 0.33
LMNA P02545 2/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
CTSD P07339 1/20 0.33
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21708670 0.83 MEN1 (0.36) KMT2AMEN1TSHRATMTAS1R3
SCHEMBL21708655 0.80 MEN1 (0.38) KMT2AMEN1TSHRATMTAS1R3
SCHEMBL9009606 0.79 NPSR1 (0.44) KMT2AMEN1TSHRATMGAA
SCHEMBL21708674 0.77 ADRB2 (0.33) KMT2AMEN1TAS1R3TAS1R1CTSS
SCHEMBL21656569 0.76 GAA (0.39) KMT2AMEN1TSHRATMGAA
SCHEMBL21632076 0.74 KMT2A (0.44) KMT2AMEN1ATMGAALMNA
SCHEMBL21708743 0.74 MEN1 (0.41) KMT2AMEN1TSHRATMTAS1R3
SCHEMBL21708649 0.73 NR3C1 (0.39) TAS1R3TAS1R1L3MBTL1
SCHEMBL21708691 0.73 LMNA (0.36) KMT2AGAALMNARAB9ASMN1; SMN2
SCHEMBL21708724 0.73 NR3C2 (0.35) TAS1R3TAS1R1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3609869-A1 SUBSTITUTED N-ARYLETHYL-2-ARYLQUINOLINE-4-CARBOXAMIDES AND USE THEREOF Bayer Aktiengesellschaft (DE) 2020-02-19 EP disclosed