SCHEMBL21708670

SCHEMBL21708670

CCCC(F)OC(=O)CC(C)(C#N)c1ccccc1OC

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
TSHR P16473 3/20 0.36
ATM Q13315 1/20 0.35
TAS1R3 Q7RTX0 1/20 0.34
TAS1R1 Q7RTX1 1/20 0.34
CTSS P25774 1/20 0.34
CTSK P43235 1/20 0.34
LMNA P02545 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
GAA P10253 2/20 0.32
RBP4 P02753 2/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
ALDH1A1 P00352 1/20 0.31
AKR1C3 P42330 1/20 0.31
AKR1C2 P52895 1/20 0.31
CYP1A2 P05177 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21708724 0.89 NR3C2 (0.35) TAS1R3TAS1R1L3MBTL1
SCHEMBL21708649 0.88 NR3C1 (0.39) TAS1R3TAS1R1L3MBTL1
SCHEMBL21708795 0.86 TAS1R3 (0.33) TAS1R3TAS1R1CTSKALDH1A1
SCHEMBL21708769 0.85 TAS1R3 (0.34) KMT2ATSHRTAS1R3TAS1R1CTSS
SCHEMBL21708762 0.83 KMT2A (0.37) MEN1KMT2ATSHRATMTAS1R3
SCHEMBL21708743 0.82 MEN1 (0.41) MEN1KMT2ATSHRATMTAS1R3
SCHEMBL21708754 0.78
SCHEMBL21656175 0.78 MTNR1A (0.41) MEN1KMT2ATSHRATMLMNA
SCHEMBL21632040 0.76 POLB (0.45) MEN1KMT2ATSHRATMLMNA
SCHEMBL21708655 0.74 MEN1 (0.38) MEN1KMT2ATSHRATMTAS1R3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3609869-A1 SUBSTITUTED N-ARYLETHYL-2-ARYLQUINOLINE-4-CARBOXAMIDES AND USE THEREOF Bayer Aktiengesellschaft (DE) 2020-02-19 EP disclosed