SCHEMBL21708902

SCHEMBL21708902

C#CCOc1cc(C(O)CN)c(C#C)cc1O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 4/20 0.35
ADRA1A P35348 4/20 0.35
ADRB2 P07550 3/20 0.35
ADRA2B P18089 3/20 0.35
ADRA2C P18825 3/20 0.35
CYP3A4 P08684 2/20 0.35
HSD17B10 Q99714 1/20 0.35
BLM P54132 4/20 0.34
MAPT P10636 3/20 0.34
APEX1 P27695 3/20 0.34
RECQL P46063 3/20 0.34
TDP1 Q9NUW8 3/20 0.34
KDM4E B2RXH2 2/20 0.34
RAD52 P43351 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
KDM4C Q9H3R0 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
NFKB1 P19838 1/20 0.33
PMP22 Q01453 1/20 0.33
CGAS Q8N884 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21708865 0.90 MAOB (0.33) ADRA2AADRA1AADRB2ADRA2BADRA2C
SCHEMBL21709245 0.85 P2RX3 (0.31) CGASP2RX3P2RX2
SCHEMBL21709249 0.83 MAOA (0.31)
SCHEMBL21708891 0.83 KDM1A (0.35) CGASMAOB
SCHEMBL21708877 0.75 HTR2A (0.39) CYP3A4HSD17B10BLMMAPTAPEX1
SCHEMBL21709056 0.75 NFKB1 (0.61) ADRA2AADRA1AADRB2ADRA2BADRA2C
SCHEMBL21709082 0.74 ADRA1A (0.49) ADRA2AADRA1ABLMNFKB1PMP22
SCHEMBL21709155 0.73 NFKB1 (0.35) ADRA2AADRA1AADRB2ADRA2BADRA2C
SCHEMBL21709247 0.72 LOXL2 (0.32) MAOBP2RX3P2RX2
SCHEMBL21708904 0.72 KDM1A (0.37) MAOBP2RX3P2RX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020032080-A1 COMPOUND, SALT OF COMPOUND, NEUROMODULATION AGENT, METHOD FOR EVALUATING NEUROMODULATION AGENT, METHOD FOR PRODUCING COMPOUND, AND METHOD FOR PRODUCING SALT OF COMPOUND 学校法人慶應義塾 2020-02-13 WO disclosed