SCHEMBL21709053

SCHEMBL21709053

C#CCNCC(O)c1ccc(OCC#C)c(OCC#C)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 2/20 0.40
ADRB2 P07550 8/20 0.40
DRD2 P14416 6/20 0.40
DRD3 P35462 6/20 0.40
DRD1 P21728 5/20 0.40
ADRB1 P08588 5/20 0.40
DRD4 P21917 4/20 0.40
HIF1A Q16665 4/20 0.39
LMNA P02545 3/20 0.39
ALDH1A1 P00352 3/20 0.39
CYP3A4 P08684 3/20 0.39
MAOA P21397 1/20 0.39
MAOB P27338 1/20 0.39
SLC22A3 O75751 1/20 0.38
SLC6A4 P31645 2/20 0.36
TSHR P16473 2/20 0.36
NPSR1 Q6W5P4 1/20 0.36
SLC22A1 O15245 1/20 0.36
CHRM2 P08172 1/20 0.36
CHRM1 P11229 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21709054 0.89 SLC22A3 (0.48) ADRB2DRD2DRD3DRD1ADRB1
SCHEMBL21709076 0.83 ADRB2 (0.52) ADRB2DRD2DRD3DRD1ADRB1
SCHEMBL21709067 0.82 KDM1A (0.34) KDM1ALMNAMAOAMAOBTSHR
SCHEMBL21708896 0.80 NFKB1 (0.49) ADRB2DRD2DRD3DRD1ADRB1
SCHEMBL21709164 0.79 KDM1A (0.35) KDM1AADRB2DRD2DRD3DRD1
SCHEMBL21709145 0.79 KDM1A (0.35) KDM1ALMNAMAOAMAOB
SCHEMBL21708904 0.77 KDM1A (0.37) KDM1AMAOAMAOB
SCHEMBL21708856 0.75 ADRB2 (0.63) ADRB2DRD2DRD3DRD1ADRB1
SCHEMBL21709065 0.74 MAOA (0.40) KDM1AADRB2DRD2DRD3DRD1
SCHEMBL16774308 0.71 PPARG (0.51) DRD2HIF1AMAOAMAOBNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020032080-A1 COMPOUND, SALT OF COMPOUND, NEUROMODULATION AGENT, METHOD FOR EVALUATING NEUROMODULATION AGENT, METHOD FOR PRODUCING COMPOUND, AND METHOD FOR PRODUCING SALT OF COMPOUND 学校法人慶應義塾 2020-02-13 WO disclosed