SCHEMBL21708865

SCHEMBL21708865

C#CCOc1cc(C#C)c(C(O)CN)cc1OCC#C

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 3/20 0.33
ADRA2A P08913 2/20 0.33
ADRA1A P35348 2/20 0.33
LOXL2 Q9Y4K0 1/20 0.33
HPGD P15428 2/20 0.32
TSHR P16473 1/20 0.32
LMNA P02545 1/20 0.32
HTR2C P28335 2/20 0.32
HTR2B P41595 2/20 0.32
HTR2A P28223 1/20 0.32
P2RX3 P56373 1/20 0.31
P2RX2 Q9UBL9 1/20 0.31
ADRB2 P07550 1/20 0.31
CYP3A4 P08684 1/20 0.31
HSD17B10 Q99714 1/20 0.31
ADRA2B P18089 1/20 0.31
ADRA2C P18825 1/20 0.31
PGK1 P00558 1/20 0.31
EGFR P00533 1/20 0.31
MAPT P10636 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21708902 0.90 ADRA2A (0.35) MAOBADRA2AADRA1AHPGDLMNA
SCHEMBL21709247 0.82 LOXL2 (0.32) MAOBLOXL2HTR2CHTR2BHTR2A
SCHEMBL21709244 0.81 MAOA (0.32)
SCHEMBL21708904 0.81 KDM1A (0.37) MAOBP2RX3P2RX2PGK1EGFR
SCHEMBL21709082 0.81 ADRA1A (0.49) ADRA2AADRA1ATSHRLMNAP2RX3
SCHEMBL21709155 0.77 NFKB1 (0.35) MAOBADRA2AADRA1AHPGDTSHR
SCHEMBL21708896 0.75 NFKB1 (0.49) MAOBADRA2AADRA1AHPGDTSHR
SCHEMBL21709245 0.75 P2RX3 (0.31) P2RX3P2RX2
SCHEMBL21709249 0.73 MAOA (0.31)
SCHEMBL21708858 0.71 HTR2A (0.42) MAOBLOXL2HTR2CHTR2BHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020032080-A1 COMPOUND, SALT OF COMPOUND, NEUROMODULATION AGENT, METHOD FOR EVALUATING NEUROMODULATION AGENT, METHOD FOR PRODUCING COMPOUND, AND METHOD FOR PRODUCING SALT OF COMPOUND 学校法人慶應義塾 2020-02-13 WO disclosed