SCHEMBL21709095

SCHEMBL21709095

C#CCn1cc(CCN)c2cc(O)cc(C#C)c21

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.31
HTR2A P28223 2/20 0.31
HTR2C P28335 2/20 0.31
HTR2B P41595 2/20 0.31
HTR3E A5X5Y0 1/20 0.31
HTR3B O95264 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C9 P11712 1/20 0.31
TSHR P16473 1/20 0.31
DRD1 P21728 1/20 0.31
HTR1D P28221 1/20 0.31
HTR1B P28222 1/20 0.31
HTR1E P28566 1/20 0.31
HTR1F P30939 1/20 0.31
HTR7 P34969 1/20 0.31
DRD3 P35462 1/20 0.31
RECQL P46063 1/20 0.31
HTR3A P46098 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21709100 0.76 MEN1 (0.33) HTR2AHTR1DRECQLMAPT
SCHEMBL21709087 0.76 EGFR (0.42) HTR1AHTR2AHTR2CHTR2BHTR3E
Hydrochloric Acid SCHEMBL21693918 0.75 EGFR (0.43) HTR1AHTR2AHTR2CHTR2BHTR3E
SCHEMBL21709093 0.67 HTR2A (0.50) HTR1AHTR2AHTR2CHTR2BHTR3E
SCHEMBL8758848 0.66 HTR2A (0.55) HTR2AHTR6MAPT
SCHEMBL21709094 0.63 TAAR1 (0.32) HTR2AHTR2CTAAR1
SCHEMBL21708941 0.62 ADRB2 (0.46) HTR1AHTR1DHTR1BHTR6MAPT
SCHEMBL28672344 0.61 HTR6 (0.46) HTR1AHTR2AHTR2CHTR2BHTR3E
SCHEMBL21708942 0.59 SPR (0.42) HTR1AHTR2CCYP1A2CYP3A4CYP2D6
SCHEMBL14801810 0.58 CHEK1 (0.37) HTR2AHTR1DHTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020032080-A1 COMPOUND, SALT OF COMPOUND, NEUROMODULATION AGENT, METHOD FOR EVALUATING NEUROMODULATION AGENT, METHOD FOR PRODUCING COMPOUND, AND METHOD FOR PRODUCING SALT OF COMPOUND 学校法人慶應義塾 2020-02-13 WO disclosed