SCHEMBL21732101

SCHEMBL21732101

CONc1cnc(N2CC(C)CC2c2cccc(F)c2)nc1

nearest known ligand 0.38

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 6/20 0.38
NTRK1 P04629 6/20 0.38
MAOB P27338 2/20 0.37
SLC6A9 P48067 7/20 0.37
MAOA P21397 1/20 0.37
RIPK1 Q13546 1/20 0.35
HTR7 P34969 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21732282 0.87 NTRK1 (0.40) JAK2NTRK1MAOBSLC6A9MAOA
SCHEMBL21732102 0.83 NTRK1 (0.44) JAK2NTRK1MAOBSLC6A9MAOA
SCHEMBL21723232 0.83 BACE1 (0.39) JAK2NTRK1MAOBSLC6A9MAOA
SCHEMBL21732277 0.81 NTRK1 (0.51) JAK2NTRK1RIPK1
SCHEMBL21732293 0.80 NTRK1 (0.46) JAK2NTRK1MAOBSLC6A9MAOA
SCHEMBL21723531 0.72 NTRK1 (0.40) JAK2NTRK1MAOBSLC6A9RIPK1
SCHEMBL21723160 0.72 HDAC1 (0.40) JAK2NTRK1MAOBSLC6A9MAOA
SCHEMBL21732197 0.69 NTRK1 (0.39) JAK2NTRK1
SCHEMBL21732073 0.68 MEN1 (0.42) JAK2NTRK1MAOBMAOA
SCHEMBL23170498 0.63 RIPK1 (0.38) MAOBMAOARIPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020035557-A1 NOVEL HETEROAROMATIC MODULATORS OF THE RETINOID-RELATED ORPHAN RECEPTOR GAMMA LEO PHARMA A/S (DK) 2020-02-20 WO disclosed