SCHEMBL21732282

SCHEMBL21732282

CONc1ccc(N2CC(C)CC2c2cccc(F)c2)nc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 10/20 0.40
JAK2 O60674 9/20 0.40
SLC6A9 P48067 3/20 0.38
HDAC1 Q13547 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
MAOB P27338 2/20 0.36
NR3C2 P08235 1/20 0.35
MAOA P21397 1/20 0.35
INSR P06213 1/20 0.35
LYN P07948 1/20 0.35
RET P07949 1/20 0.35
MET P08581 1/20 0.35
ROS1 P08922 1/20 0.35
FGR P09769 1/20 0.35
KIT P10721 1/20 0.35
FGFR4 P22455 1/20 0.35
FGFR3 P22607 1/20 0.35
TIE1 P35590 1/20 0.35
KDR P35968 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21732101 0.87 JAK2 (0.38) NTRK1JAK2SLC6A9MAOBMAOA
SCHEMBL21723531 0.82 NTRK1 (0.40) NTRK1JAK2SLC6A9HDAC1HDAC8
SCHEMBL21723160 0.81 HDAC1 (0.40) NTRK1JAK2SLC6A9HDAC1HDAC8
SCHEMBL21732284 0.73 RORC (0.49) NTRK1JAK2
SCHEMBL21732102 0.73 NTRK1 (0.44) NTRK1JAK2SLC6A9MAOBMAOA
SCHEMBL21723232 0.72 BACE1 (0.39) NTRK1JAK2SLC6A9MAOBMAOA
SCHEMBL21732277 0.71 NTRK1 (0.51) NTRK1JAK2INSRLYNRET
SCHEMBL21732293 0.69 NTRK1 (0.46) NTRK1JAK2SLC6A9MAOBMAOA
SCHEMBL21732201 0.69 HDAC6 (0.44) NTRK1HDAC1HDAC8HDAC6MAOB
SCHEMBL23170498 0.62 RIPK1 (0.38) MAOBMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020035557-A1 NOVEL HETEROAROMATIC MODULATORS OF THE RETINOID-RELATED ORPHAN RECEPTOR GAMMA LEO PHARMA A/S (DK) 2020-02-20 WO disclosed