SCHEMBL2174563

SCHEMBL2174563

COC(=O)c1ccc(O)c2ccccc12

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.61
LMNA P02545 3/20 0.60
TSHR P16473 1/20 0.60
CA1 P00915 4/20 0.52
CA2 P00918 4/20 0.52
CA9 Q16790 4/20 0.52
CA12 O43570 3/20 0.52
CA7 P43166 3/20 0.52
CA14 Q9ULX7 3/20 0.52
PDK2 Q15119 1/20 0.52
PDK4 Q16654 1/20 0.52
BRD4 O60885 2/20 0.51
MEN1 O00255 1/20 0.51
MAPT P10636 1/20 0.51
KMT2A Q03164 1/20 0.51
NR4A2 P43354 2/20 0.50
IDO1 P14902 1/20 0.50
CREBBP Q92793 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.49
GAA P10253 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29434198 0.90 BRD4 (0.59) KDM4ELMNATSHRCA1CA2
SCHEMBL70381 0.90 BRD4 (0.59) KDM4ELMNATSHRCA1CA2
SCHEMBL9300933 0.89 LMNA (0.66) KDM4ELMNATSHRCA1CA2
SCHEMBL9166724 0.84 IDO1 (0.54) KDM4ELMNATSHRMEN1MAPT
SCHEMBL982076 0.82 BRD4 (0.53) KDM4ELMNATSHRBRD4MEN1
SCHEMBL5750893 0.82 BRD4 (0.53) KDM4ELMNATSHRBRD4MEN1
SCHEMBL31049726 0.82 BRD4 (0.53) KDM4ELMNATSHRBRD4MEN1
SCHEMBL31049722 0.82 BRD4 (0.53) KDM4ELMNATSHRBRD4MEN1
SCHEMBL1600050 0.81 IDO1 (0.46) KDM4ELMNATSHRMEN1MAPT
SCHEMBL70429 0.81 LMNA (0.59) KDM4ELMNATSHRCA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 38 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119136797-A CB1Ligand conjugated compounds and uses thereof 阿达尔克斯制药有限公司 2024-12-13 CN disclosed
CN-118307518-A Polycyclic PARP selective inhibitors 轩竹生物科技股份有限公司 2024-07-09 CN disclosed
CN-111936499-B Heterobicyclic inhibitors of MAT2A and methods for treating cancer 法国施维雅药厂 2023-09-19 CN disclosed
WO-2023168296-A2 CB1 LIGAND CONJUGATED COMPOUNDS AND USES THEREOF ADARX PHARMACEUTICALS, INC. (US) 2023-09-07 WO disclosed
US-20160289160-A1 PRODUCTION METHOD FOR ARYL (METH) ACRYLATE MITSUBISHI RAYON CO., LTD. (JP) 2016-10-06 US disclosed
EP-2977367-A1 PRODUCTION METHOD FOR (METH) ACRYLATE ARYL ESTER Mitsubishi Rayon Co., Ltd. (JP) 2016-01-27 EP disclosed
CN-105051000-A Process for producing aryl (meth) acrylate MITSUBISHI RAYON CO 2015-11-11 CN disclosed
CN-103827121-A oxy-cyclohexyl-4H, 6H-5-oxa-2, 3,10 b-triaza-benzo [ e ] azulenes as V1a antagonists HOFFMANN LA ROCHE 2014-05-28 CN disclosed
CN-101772506-B Macrocycles and their uses NOVARTIS AG 2014-02-12 CN disclosed
US-8642629-B2 Naphthylacetic acids HOFFMANN-LA ROCHE INC. (US) 2014-02-04 US disclosed
EP-1546086-A2 AMINOALCOHOL DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2005-06-29 EP disclosed
US-20040006143-A1 For therapy of urinary incontinence FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-01-08 US disclosed
WO-2004002939-A2 AMINOALCOHOL DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-01-08 WO disclosed
US-6613942-B1 Nonpeptide; 4-hydroxy benzoic acid hydrazides NOVO NORDISK A/S (DK) 2003-09-02 US disclosed
CN-1267281-A Glucagon antagonists/inverse agonists NOVO NORDISK AS (DK) 2000-09-20 CN disclosed
EP-0994848-A1 GLUCAGON ANTAGONISTS/INVERSE AGONISTS NOVO NORDISK A/S (DK) 2000-04-26 EP disclosed
WO-1999001423-A1 GLUCAGON ANTAGONISTS/INVERSE AGONISTS NOVO NORDISK A/S (DK) 1999-01-14 WO disclosed
WO-1999001423-A1 GLUCAGON ANTAGONISTS/INVERSE AGONISTS NOVO NORDISK A/S (DK) 1999-01-14 WO disclosed
US-5298593-A Polymerization of ester monomer, aromatic dicarboxylic acid, and oxyaromatic carboxylic acid MITSUBISHI PETROCHEMICAL COMPANY, LTD. (JP) 1994-03-29 US disclosed
EP-0520428-A2 Method of producing thermotropic liquid crystalline polyester MITSUBISHI CHEMICAL CORPORATION (JP) 1992-12-30 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160289160-A1 PRODUCTION METHOD FOR ARYL (METH) ACRYLATE ACR, ALK, GNPAT KDM4E 677/4885LMNA 4763/4885TSHR 405/4885
US-20040006143-A1 For therapy of urinary incontinence H1-0, HRH2, H1-2 KDM4E 1554/4885LMNA 4565/4885TSHR 3005/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.