SCHEMBL21746470

SCHEMBL21746470

CN/C=C\C(=N)c1ccc(O)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 7/20 0.40
MAPT P10636 6/20 0.40
LMNA P02545 4/20 0.40
KMT2A Q03164 3/20 0.40
HSD17B10 Q99714 3/20 0.40
MEN1 O00255 2/20 0.40
NR3C1 P04150 2/20 0.40
TP53 P04637 2/20 0.40
CYP1A2 P05177 2/20 0.40
CYP3A4 P08684 2/20 0.40
ADORA3 P0DMS8 2/20 0.40
CYP2D6 P10635 2/20 0.40
CYP2C9 P11712 2/20 0.40
ALOX15 P16050 2/20 0.40
CYP2C19 P33261 2/20 0.40
OPRD1 P41143 2/20 0.40
HIF1A Q16665 2/20 0.40
GAA P10253 1/20 0.40
ALOX12 P18054 1/20 0.40
CA12 O43570 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13874287 0.84 ALDH1A1 (0.42) MAPTLMNAKMT2AMEN1HIF1A
SCHEMBL14141387 0.82 PKM (0.38) MAPTLMNAKMT2AHSD17B10MEN1
SCHEMBL21746252 0.79 PRSS1 (0.48) MAPTKMT2AMEN1CYP3A4CA1
SCHEMBL19443447 0.78 LOXL2 (0.48) ABAT
SCHEMBL14204477 0.78 MAPT (0.42) MAPTLMNAKMT2AHSD17B10MEN1
SCHEMBL18871578 0.77 ESR1 (0.39) ESR1MAPTKMT2AHSD17B10MEN1
SCHEMBL21746584 0.75 HDAC3 (0.42) ALDH1A1TSHR
SCHEMBL18831458 0.75 HSP90AA1 (0.40) MAPTLMNAKMT2AHSD17B10MEN1
SCHEMBL17267202 0.74 HDAC1 (0.46) MAPTLMNAKMT2AMEN1CYP1A2
SCHEMBL21746596 0.74 ELANE (0.47) ESR1MAPTLMNAKMT2AHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2944637-B1 NITROGEN-CONTAINING HETEROCYLIC COMPOUND OR SALT THEREOF FUJIFILM CORP (JP) 2020-02-19 EP disclosed