SCHEMBL21746252

SCHEMBL21746252

CN/C=C\C(=N)c1ccc(OC)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRSS1 P07477 1/20 0.48
PRSS2 P07478 1/20 0.48
PRSS3 P35030 1/20 0.48
PLK1 P53350 1/20 0.46
CA1 P00915 4/20 0.44
CA2 P00918 4/20 0.44
CES2 O00748 1/20 0.42
CES1 P23141 1/20 0.42
ALDH1A1 P00352 4/20 0.42
MAPT P10636 3/20 0.42
KDM4E B2RXH2 2/20 0.42
HPGD P15428 2/20 0.42
CYP3A4 P08684 1/20 0.41
F3 P13726 1/20 0.41
PTGIR P43119 1/20 0.41
HDAC3 O15379 1/20 0.41
HDAC4 P56524 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC7 Q8WUI4 1/20 0.41
HDAC2 Q92769 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21746596 0.80 ELANE (0.47) ALDH1A1MAPTKDM4ECYP3A4SMN1; SMN2
SCHEMBL21745729 0.80 PRSS1 (0.54) PRSS1PRSS2PRSS3CES2CES1
SCHEMBL13874287 0.79 ALDH1A1 (0.42) CES2CES1ALDH1A1MAPTKDM4E
SCHEMBL21746470 0.79 ESR1 (0.40) CA1CA2ALDH1A1MAPTHPGD
SCHEMBL21746471 0.79 NR1I2 (0.49) PRSS1PLK1ALDH1A1MAPTCYP3A4
SCHEMBL8294719 0.78 PRSS1 (0.57) PRSS1PRSS2PRSS3CA1CA2
SCHEMBL14141387 0.77 PKM (0.38) PRSS1PRSS2PRSS3ALDH1A1MAPT
SCHEMBL18871269 0.76 ALOX15 (0.43) ALDH1A1MAPTKDM4ESMN1; SMN2MEN1
SCHEMBL18831379 0.74 ALDH1A1 (0.51) ALDH1A1MAPTKDM4EHPGDCYP3A4
SCHEMBL28480552 0.73 PRSS1 (0.55) PRSS1PRSS2PRSS3CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2944637-B1 NITROGEN-CONTAINING HETEROCYLIC COMPOUND OR SALT THEREOF FUJIFILM CORP (JP) 2020-02-19 EP disclosed