SCHEMBL21747477

SCHEMBL21747477

O=C(Nc1ccccc1-c1nc2cc(CN3CCN(C(=O)O)CC3)ccc2o1)c1cnc2ccccc2n1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT1 Q96EB6 3/20 0.51
CHRM2 P08172 1/20 0.45
ADRA2A P08913 1/20 0.45
CHRM1 P11229 1/20 0.45
SLC6A2 P23975 1/20 0.45
SIRT2 Q8IXJ6 1/20 0.45
SIRT3 Q9NTG7 1/20 0.45
FAAH O00519 7/20 0.44
ACKR3 P25106 1/20 0.43
S1PR1 P21453 1/20 0.42
S1PR3 Q99500 1/20 0.42
HSD17B10 Q99714 2/20 0.42
BCHE P06276 2/20 0.41
HDAC6 Q9UBN7 1/20 0.41
KDM4E B2RXH2 1/20 0.40
NPC1 O15118 1/20 0.40
ALDH1A1 P00352 1/20 0.40
TP53 P04637 1/20 0.40
POLB P06746 1/20 0.40
HPGD P15428 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21747442 0.91 SIRT1 (0.52) SIRT1CHRM2ADRA2ACHRM1SLC6A2
SCHEMBL30468245 0.89 SIRT1 (0.64) SIRT1CHRM2ADRA2ACHRM1SLC6A2
SCHEMBL21747481 0.88 SIRT1 (0.49) SIRT1CHRM2ADRA2ACHRM1SLC6A2
SCHEMBL21747469 0.87 HSD17B10 (0.48) S1PR1S1PR3HSD17B10BCHEHDAC6
Trifluoroacetic Acid SCHEMBL21747462 0.86 SIRT1 (0.59) SIRT1CHRM2ADRA2ACHRM1SLC6A2
SCHEMBL21747446 0.84 TP53 (0.49) FAAHS1PR1S1PR3HSD17B10BCHE
SCHEMBL21747494 0.80 HSD17B10 (0.57) SIRT1HSD17B10KDM4ENPC1ALDH1A1
SCHEMBL21747471 0.79 HDAC1 (0.50) S1PR1S1PR3HSD17B10HDAC6KDM4E
SCHEMBL21747444 0.78 S1PR1 (0.50) S1PR1S1PR3HDAC6NPC1RAB9A
SCHEMBL21747493 0.77 SIRT1 (0.51) SIRT1S1PR1S1PR3HSD17B10HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3613735-A1 NOVEL SIRT 1 ACTIVATOR AND MEDICINAL USE THEREOF Pusan National University Industry - University Cooperation Foundation (KR) 2020-02-26 EP disclosed