SCHEMBL21756936

SCHEMBL21756936

CC(C)c1c(F)cc(I)cc1CN1CCOCC1

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP2A13 Q16696 7/20 0.47
MAPT P10636 1/20 0.43
KCNH2 Q12809 6/20 0.41
CYP2C9 P11712 1/20 0.40
ALOX15 P16050 1/20 0.40
HSD17B10 Q99714 1/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
POLB P06746 1/20 0.38
NPSR1 Q6W5P4 1/20 0.37
CNR2 P34972 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21769976 0.81 CYP2A13 (0.50) CYP2A13CYP2C9ALOX15HSD17B10MEN1
SCHEMBL26812028 0.76 CYP2A13 (0.40) CYP2A13MAPTKCNH2CYP2C9ALOX15
SCHEMBL15546497 0.75 CYP2A13 (0.61) CYP2A13MAPTCYP2C9ALOX15HSD17B10
SCHEMBL21756943 0.74 MAPT (0.51) CYP2A13MAPTKCNH2CYP2C9ALOX15
SCHEMBL26812751 0.73 PIK3C3 (0.41) CYP2A13MAPTKCNH2
SCHEMBL13091284 0.71 KCNH2 (0.57) CYP2A13MAPTKCNH2CYP2C9ALOX15
SCHEMBL21756947 0.71 SLC6A4 (0.32) KCNH2
SCHEMBL21756927 0.71 GABRA1 (0.31)
SCHEMBL21756926 0.71 GABRA1 (0.35)
SCHEMBL21756924 0.69 GABRA1 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020039092-A2 NOVEL AROMATIC MOLECULES Xeniopro GmbH (DE) 2020-02-27 WO disclosed
WO-2020039094-A1 PHENOXY(HETERO)ARYL ETHERS OF ANTIPROLIFERATIVE ACTIVITY Xeniopro GmbH (DE) 2020-02-27 WO disclosed
US-9403829-B2 Pharmaceutical compositions of 7-(6-(2-hydroxypropan-2-yl)pyridin-3-yl)-1-((trans)-4-methoxycyclohexyl)-3,4-dihydropyrazino [2,3-b]pyrazin-2(1H)-one, a solid form thereof and methods of their use SIGNAL PHARMACEUTICALS, LLC (US) 2016-08-02 US disclosed