SCHEMBL21770489

SCHEMBL21770489

CSc1ccc(-c2ccc(CO)nc2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 1/20 0.42
PI4KA P42356 1/20 0.42
PI4KB Q9UBF8 1/20 0.42
MAOB P27338 1/20 0.38
HAO1 Q9UJM8 1/20 0.38
S1PR1 P21453 1/20 0.37
TLR9 Q9NR96 1/20 0.37
TLR8 Q9NR97 1/20 0.37
TLR7 Q9NYK1 1/20 0.37
KDM5B Q9UGL1 1/20 0.35
GSK3B P49841 1/20 0.35
DYRK1A Q13627 1/20 0.35
SLC6A4 P31645 1/20 0.35
MMP12 P39900 1/20 0.35
MMP13 P45452 1/20 0.35
NPC1 O15118 1/20 0.35
LMNA P02545 1/20 0.35
TP53 P04637 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2658413 0.85 MBOAT4 (0.40) PIK3CAPI4KAPI4KBS1PR1SLC6A4
SCHEMBL29694695 0.85 MBOAT4 (0.40) PIK3CAPI4KAPI4KBS1PR1SLC6A4
SCHEMBL21769960 0.82 MAOB (0.38) MAOBHAO1SLC6A4MMP12MMP13
SCHEMBL5114909 0.77 PIK3CA (0.46) PIK3CAPI4KAPI4KBNPC1RAB9A
SCHEMBL22920103 0.76 PIK3CA (0.45) PIK3CAPI4KAPI4KBS1PR1TLR9
SCHEMBL6879617 0.76 NOTUM (0.47) PIK3CAPI4KAPI4KBNPC1RAB9A
SCHEMBL4212545 0.73 MAOB (0.42) MAOBHAO1NPC1LMNARAB9A
SCHEMBL8423018 0.72 PTGS2 (0.51) PIK3CAPI4KB
SCHEMBL4415453 0.71 KIF11 (0.47) PIK3CAPI4KAPI4KBMAOBDYRK1A
SCHEMBL10300271 0.71 ALDH1A1 (0.50) HAO1SLC6A4MMP12MMP13NISCH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020039027-A1 PYRROLIDINE GLYCOSIDASE INHIBITORS ASCENEURON S. A. (CH) 2020-02-27 WO disclosed