SCHEMBL2178905

SCHEMBL2178905

O=S(=O)(c1ccc(C(Oc2cncc(Cl)c2)c2cc3ncc(Cl)nc3[nH]2)cc1)C1CC1

nearest known ligand 0.38

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GCK P35557 9/20 0.38
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
CCR2 P41597 1/20 0.32
EPAS1 Q99814 1/20 0.31
NAMPT P43490 1/20 0.31
CNR1 P21554 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2179681 0.82 GCK (0.48) GCK
SCHEMBL2365130 0.77 GCK (0.35) GCKNAMPT
SCHEMBL2178177 0.75 GCK (0.47) GCK
SCHEMBL2177869 0.69 GCK (0.44) GCK
SCHEMBL2178179 0.69 ALDH1A1 (0.34) GCKNAMPTCNR1
SCHEMBL2180026 0.68 GCK (0.48) GCK
SCHEMBL2179805 0.67 CNR2 (0.38) GCKCYP3A4
SCHEMBL2178624 0.67 GCK (0.38) GCKCNR1
SCHEMBL2197573 0.66 PIK3CA (0.34) GCK
SCHEMBL2198311 0.64 GCK (0.60) GCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011080755-A1 FUSED NITROGEN HETEROCYCLIC COMPOUNDS, PROCESS OF PREPARATION AND USES THEREOF ADVINUS THERAPEUTICS PRIVATE LIMITED (IN) 2011-07-07 WO claimed
WO-2011080755-A1 FUSED NITROGEN HETEROCYCLIC COMPOUNDS, PROCESS OF PREPARATION AND USES THEREOF ADVINUS THERAPEUTICS PRIVATE LIMITED (IN) 2011-07-07 WO disclosed