SCHEMBL21789147

SCHEMBL21789147

COC(=O)[Si@@H](NCc1ccc(C(F)(F)F)cc1)C1CCC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.43
MAPT P10636 1/20 0.43
MAPK1 P28482 1/20 0.43
P2RX7 Q99572 1/20 0.41
KCNH2 Q12809 2/20 0.41
HRH3 Q9Y5N1 1/20 0.41
TEAD1 P28347 1/20 0.40
LSS P48449 1/20 0.40
SCN9A Q15858 1/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
SRD5A2 P31213 1/20 0.39
KCNQ3 O43525 1/20 0.39
KCNQ2 O43526 1/20 0.39
KCNQ4 P56696 1/20 0.39
KCNQ5 Q9NR82 1/20 0.39
MAPK14 Q16539 1/20 0.38
FFAR1 O14842 1/20 0.38
MTOR P42345 1/20 0.38
PPARA Q07869 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21865601 0.73 P2RX7 (0.42) CYP3A4MAPTMAPK1P2RX7KCNH2
SCHEMBL4481286 0.71 CCR2 (0.47) CYP3A4MAPTMAPK1P2RX7TEAD1
SCHEMBL21789150 0.71 ITGB3 (0.45) CYP3A4MAPTMAPK1P2RX7KCNH2
SCHEMBL4495364 0.71 CCR2 (0.47) CYP3A4MAPTMAPK1P2RX7TEAD1
SCHEMBL21865730 0.71 ITGB3 (0.45) CYP3A4MAPTMAPK1P2RX7KCNH2
SCHEMBL26154086 0.70 ALDH1A1 (0.65) MAPTP2RX7KCNH2HRH3ALDH1A1
SCHEMBL21777493 0.68 TPSAB1 (0.50) P2RX7KCNH2HRH3TEAD1LSS
SCHEMBL16839732 0.67 OPRL1 (0.41) LSSMAPK14FFAR1MTORPPARA
SCHEMBL16839734 0.67 OPRL1 (0.41) LSSMAPK14FFAR1MTORPPARA
SCHEMBL19650799 0.67 BCHE (0.61) HRH3TEAD1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020047447-A1 CARDIAC SARCOMERE INHIBITORS CYTOKINETICS, INC. (US) 2020-03-05 WO disclosed