SCHEMBL21798462

SCHEMBL21798462

CNC(=O)O[C@H]1CCOc2ccccc21

nearest known ligand 0.50

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SSTR4 P31391 1/20 0.41
BCHE P06276 2/20 0.39
MAPK1 P28482 2/20 0.37
ACHE P22303 3/20 0.36
TRPV1 Q8NER1 4/20 0.36
BRD4 O60885 2/20 0.36
CREBBP Q92793 2/20 0.36
KMT2A Q03164 1/20 0.36
KDM4E B2RXH2 1/20 0.36
XIAP P98170 1/20 0.36
GAA P10253 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29208044 0.85 SSTR4 (0.46) SSTR4MAPK1TRPV1BRD4CREBBP
SCHEMBL30812977 0.84 POLB (0.44) SSTR4MAPK1TRPV1KDM4EGAA
SCHEMBL9785817 0.84 POLB (0.44) SSTR4MAPK1TRPV1KDM4EGAA
SCHEMBL7300865 0.81 SSTR4 (0.42) SSTR4MAPK1TRPV1BRD4CREBBP
SCHEMBL24262284 0.79 SSTR4 (0.38) SSTR4MAPK1BRD4CREBBPKDM4E
SCHEMBL27720908 0.78 SSTR4 (0.40) SSTR4MAPK1KMT2AGAASMN1; SMN2
SCHEMBL2740802 0.76 SSTR4 (0.41) SSTR4MAPK1KMT2AKDM4EGAA
SCHEMBL27346326 0.76 SSTR4 (0.46) SSTR4KMT2AGAA
SCHEMBL13444800 0.75 ITGB2 (0.41) SSTR4MAPK1SMN1; SMN2
SCHEMBL2583594 0.75 BCHE (0.39) BCHEMAPK1ACHEGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10738064-B2 Chiral α-amino tertiary boronic esters PURDUE RESEARCH FOUNDATION (US) 2020-08-11 US disclosed
US-20200079799-A1 Novel Chiral Alfa-Amino Tertiary Boronic Esters PURDUE RESEARCH FOUNDATION (US) 2020-03-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200079799-A1 Novel Chiral Alfa-Amino Tertiary Boronic Esters HBB, BCAT1, BCAT2 SSTR4 218/4885BCHE 11/4885MAPK1 3580/4885
US-10738064-B2 Chiral α-amino tertiary boronic esters HBB, BCAT1, BCAT2 SSTR4 167/4885BCHE 11/4885MAPK1 3000/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.