SCHEMBL2179945

SCHEMBL2179945

C=CCC(O)(C(C)=O)C(=O)O

nearest known ligand 0.38

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.38
TSHR P16473 2/20 0.38
HTT P42858 1/20 0.32
MAPT P10636 1/20 0.31
TET2 Q6N021 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29039008 1.00 ALDH1A1 (0.38) ALDH1A1TSHRHTTMAPTTET2
SCHEMBL28648606 1.00 ALDH1A1 (0.38) ALDH1A1TSHRHTTMAPTTET2
SCHEMBL27776897 0.88 ALDH1A1 (0.36) ALDH1A1TSHRHTTMAPT
SCHEMBL10773383 0.85 ALDH1A1 (0.43) ALDH1A1TSHRHTTMAPTTET2
SCHEMBL5998401 0.78 MAPT (0.42) ALDH1A1TSHRMAPT
SCHEMBL5998393 0.78 MAPT (0.42) ALDH1A1TSHRMAPT
Acetic Acid SCHEMBL8947198 0.77 TET2 (0.43) ALDH1A1TSHRHTTMAPTTET2
SCHEMBL5998397 0.77 ALDH1A1 (0.35) ALDH1A1TSHRHTT
SCHEMBL30513348 0.76
SCHEMBL3256852 0.76

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114805068-B Preparation method of chiral alpha-hydroxy-beta-keto ester compound 南京工业大学 2023-07-21 CN disclosed
CN-113549062-B Chiral quaternary ammonium salt phase transfer catalyst with high steric hindrance derived from cinchona alkaloid and synthesis method thereof 南京工业大学 2022-08-09 CN disclosed
CN-114805068-A Preparation method of chiral alpha-hydroxy-beta-keto ester compound 南京工业大学 2022-07-29 CN disclosed
CN-113563187-A Preparation method of chiral alpha-hydroxy-beta-keto ester compound 南京工业大学 2021-10-29 CN disclosed
CN-113549062-A Chiral quaternary ammonium salt phase transfer catalyst with high steric hindrance derived from cinchona alkaloid and synthesis method thereof 南京工业大学 2021-10-26 CN disclosed
US-10053396-B2 Process for the specific isotopic labeling of methyl groups of Val, Leu and Ile COMMISSARIAT A L'ENERGIE ATOMIQUE ET AUX ENERGIES ALTERNATIVES (FR) 2018-08-21 US disclosed
US-20170275216-A1 PROCESS FOR THE SPECIFIC ISOTOPIC LABELING OF METHYL GROUPS OF VAL, LEU AND ILE COMMISSARIAT A L'ENERGIE ATOMIQUE ET AUX ENERGIES ALTERNATIVES (FR) 2017-09-28 US disclosed
US-9708228-B2 Process for the specific isotopic labeling of methyl groups of Val, Leu and Ile COMMISSARIAT A L'ENERGIE ATOMIQUE ET AUX ENERGIES ALTERNATIVES (FR) 2017-07-18 US disclosed
US-9708228-B2 Process for the specific isotopic labeling of methyl groups of Val, Leu and Ile COMMISSARIAT A L'ENERGIE ATOMIQUE ET AUX ENERGIES ALTERNATIVES (FR) 2017-07-18 US disclosed
EP-2521704-B1 PROCESS FOR THE SPECIFIC ISOTOPIC LABELING OF METHYL GROUPS OF VAL, LEU AND ILE COMMISSARIAT L ENERGIE ATOMIQUE ET AUX ENERGIES ALTERNATIVES (FR) 2015-09-30 EP disclosed
WO-2014024151-A1 LABELED CHIRAL ALPHA-HYDROXY KETOACID DERIVATIVES, A PROCESS FOR PREPARING SAID DERIVATIVES AND THEIR USE COMMISSARIAT A L'ENERGIE ATOMIQUE ET AUX ENERGIES ALTERNATIVES (FR) 2014-02-13 WO disclosed
US-20130122598-A1 PROCESS FOR THE SPECIFIC ISOTOPIC LABELING OF METHYL GROUPS OF VAL, LEU AND ILE COMMISSARIAT A L'ENERGIE ATOMIQUE ET AUX ENERGIES ALTERNATIVES (FR) 2013-05-16 US disclosed
US-20130122598-A1 PROCESS FOR THE SPECIFIC ISOTOPIC LABELING OF METHYL GROUPS OF VAL, LEU AND ILE COMMISSARIAT A L'ENERGIE ATOMIQUE ET AUX ENERGIES ALTERNATIVES (FR) 2013-05-16 US disclosed
EP-2521704-A1 PROCESS FOR THE SPECIFIC ISOTOPIC LABELING OF METHYL GROUPS OF VAL, LEU AND ILE Commissariat à l'Énergie Atomique et aux Énergies Alternatives (FR) 2012-11-14 EP disclosed
EP-2521704-A1 PROCESS FOR THE SPECIFIC ISOTOPIC LABELING OF METHYL GROUPS OF VAL, LEU AND ILE Commissariat à l'Énergie Atomique et aux Énergies Alternatives (FR) 2012-11-14 EP disclosed
WO-2011083356-A1 PROCESS FOR THE SPECIFIC ISOTOPIC LABELING OF METHYL GROUPS OF VAL, LEU AND ILE COMMISSARIAT A L'ENERGIE ATOMIQUE ET AUX ENERGIES ALTERNATIVES (FR) 2011-07-14 WO disclosed
WO-2011083356-A1 PROCESS FOR THE SPECIFIC ISOTOPIC LABELING OF METHYL GROUPS OF VAL, LEU AND ILE COMMISSARIAT A L'ENERGIE ATOMIQUE ET AUX ENERGIES ALTERNATIVES (FR) 2011-07-14 WO disclosed
EP-1818336-A1 2,2-bis-(4-hydroxyphenyl)-alkyl onium salt and a process for the preparation thereof Council of Scientific and Industrial Research (IN) 2007-08-15 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10053396-B2 Process for the specific isotopic labeling of methyl groups of Val, Leu and Ile BCAT1, BCAT2, ALAD ALDH1A1 4057/4885TSHR 4559/4885HTT 3701/4885
US-20130122598-A1 PROCESS FOR THE SPECIFIC ISOTOPIC LABELING OF METHYL GROUPS OF VAL, LEU AND ILE BCAT1, BCAT2, SLC1A5 ALDH1A1 4604/4885TSHR 4484/4885HTT 758/4885
US-20170275216-A1 PROCESS FOR THE SPECIFIC ISOTOPIC LABELING OF METHYL GROUPS OF VAL, LEU AND ILE BCAT1, BCAT2, ALAD ALDH1A1 4057/4885TSHR 4559/4885HTT 3701/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.