Metahexamide

Metahexamide

SCHEMBL218071

Cc1ccc(S(=O)(=O)NC(=O)NC2CCCCC2)cc1N

nearest known ligand 0.68

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.68
ALDH1A1 P00352 4/20 0.62
LMNA P02545 3/20 0.62
TSHR P16473 2/20 0.62
BLM P54132 2/20 0.62
TDP1 Q9NUW8 2/20 0.62
THRB P10828 1/20 0.62
PPARG P37231 3/20 0.50
MAPT P10636 2/20 0.50
GAA P10253 1/20 0.50
KCNH2 Q12809 1/20 0.50
SMN1; SMN2 Q16637 2/20 0.49
NPC1 O15118 1/20 0.49
RAB9A P51151 1/20 0.49
HRH3 Q9Y5N1 3/20 0.48
CYP3A4 P08684 2/20 0.48
CYP2C9 P11712 2/20 0.48
CYP2C19 P33261 2/20 0.48
HTR1A P08908 1/20 0.48
NFKB1 P19838 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Metahexamide SCHEMBL30107709 1.00 ADORA3 (0.68) ADORA3ALDH1A1LMNATSHRBLM
Metahexamide SCHEMBL15845574 0.85 ADORA3 (0.62) ADORA3ALDH1A1LMNATSHRBLM
Gliclazide SCHEMBL13723694 0.85 ALDH1A1 (0.67) ADORA3ALDH1A1LMNATSHRBLM
SCHEMBL23736042 0.81 ADORA3 (0.74) ADORA3ALDH1A1LMNATSHRBLM
Glycyclamide SCHEMBL49386 0.81 ADORA3 (1.00) ADORA3ALDH1A1LMNATSHRBLM
Heptolamide SCHEMBL1814750 0.81 ADORA3 (1.00) ADORA3ALDH1A1LMNATSHRBLM
Glyoctamide SCHEMBL667731 0.81 ADORA3 (1.00) ADORA3ALDH1A1LMNATSHRBLM
Glycyclamide SCHEMBL21722119 0.80 ADORA3 (0.97) ADORA3ALDH1A1LMNATSHRBLM
Hydrochloric Acid SCHEMBL9796358 0.80 ALDH1A1 (0.71) ALDH1A1LMNATSHRTDP1GAA
Tolpentamide SCHEMBL2109411 0.80 ADORA3 (0.97) ADORA3ALDH1A1LMNATSHRBLM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 904 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4232448-A1 AGONISTS OF FREE FATTY ACID RECEPTOR 1 AND THEIR USE IN DISEASES ASSOCIATED WITH SAID RECEPTOR Halo Therapeutics Ltd (GB) 2023-08-30 EP claimed
US-20220184070-A1 LOW-DOSE TRIPLE COMBINATION FORMULATION The George Institute for Global Health (AU) 2022-06-16 US claimed
WO-2022083853-A1 AGONISTS OF FREE FATTY ACID RECEPTOR 1 AND THEIR USE IN DISEASES ASSOCIATED WITH SAID RECEPTOR GBIOTECH S.À.R.L. (CH) 2022-04-28 WO claimed
EP-3946343-A1 LOW-DOSE TRIPLE COMBINATION FORMULATION The George Institute For Global Health (AU) 2022-02-09 EP claimed
US-11213508-B2 Compositions comprising urolithins and uses thereof for the stimulation of insulin secretion UNIVERSITE DE MONTPELLIER (FR) 2022-01-04 US claimed
EP-3833336-A1 METHODS FOR DELAYING OCCURRENCE OF NEW-ONSET TYPE 2 DIABETES AND FOR SLOWING PROGRESSION OF AND TREATING TYPE 2 DIABETES DalCor Pharma UK Ltd Leatherhead, Zug Branch (CH) 2021-06-16 EP claimed
EP-2459227-B1 Prodrugs containing an aromatic amine connected by an amide bond to a carrier ASCENDIS PHARMA AS (DK) 2021-03-17 EP claimed
WO-2020194046-A1 LOW-DOSE TRIPLE COMBINATION FORMULATION The George Institute for Global Health (AU) 2020-10-01 WO claimed
CN-111201022-A Use of gaboxadol for treating diabetes and related conditions 奥维德医疗公司 2020-05-26 CN claimed
US-20200155504-A1 COMPOSITIONS COMPRISING UROLITHINS AND USES THEREOF FOR THE STIMULATION OF INSULIN SECRETION CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2020-05-21 US claimed
CN-1250226-C Combination comprising -2-ethoxy-3- [4- (2- { 4-methanesulfonyloxyphenyl } ethoxy) phenyl ] propanoic acid or 3- {4- [2- (4-tert-butoxycarbonylaminophenyl) ethoxy ] phenyl } - -2-ethoxypropanoic acid and a sulfonylurea ASTRAZENECA AB (SE) 2006-04-12 CN claimed
CN-1212117-C Pharmaceutical composition for treating diabetes TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2005-07-27 CN claimed
CN-1599612-A Combination of FBP enzyme inhibitor and antidiabetic agent for treating diabetes METABASIS THERAPEUTICS INC (US) 2005-03-23 CN claimed
CN-1537008-A Combination comprising -2-ethoxy-3- [ 4- (2- { 4-methanesulfonyloxyphenyl } ethoxy) phenyl ] propanoic acid or 3- { 4- [ 2- (4-tert-butoxycarbonylaminophenyl) ethoxy ] phenyl } - -2-ethoxypropanoic acid and a sulfonylurea 2004-10-13 CN claimed
US-20040068005-A1 Pharmaceutical combinations KERI PHARMA GENERICS KFT. (HU) 2004-04-08 US claimed
EP-1303304-A2 PHARMACEUTICAL COMBINATIONS FOR TREATMENT AND PREVENTION OF DIABETES MELLITUS Keri Pharma KFT (HU) 2003-04-23 EP claimed
CN-1400908-A Combinations comprising dipeptidyl peptidase-IV inhibitors NOVARTIS AG (CH) 2003-03-05 CN claimed
WO-2002005795-A2 PHARMACEUTICAL COMBINATIONS FOR TREATMENT AND PREVENTION OF DIABETES MELLITUS Kéri Pharma Kft. (HU) 2002-01-24 WO claimed
CN-1294519-A Pharmaceutical composition containing a compound having an activity of promoting the absorption of an active ingredient INPHARMA SA (CH) 2001-05-09 CN claimed
CN-1264303-A Treatment of diabetes with thiazolidinediones, insulin secretagogues and biguanides SMITHKLINE BEECHAM PLC (GB) 2000-08-23 CN claimed