SCHEMBL21836003

SCHEMBL21836003

c1ccc(CON2CCC2c2ccccc2)cc1

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.40
CHRNB4 P30926 1/20 0.40
CHRNA3 P32297 1/20 0.40
CHRNA7 P36544 1/20 0.40
CHRNA4 P43681 1/20 0.40
RIPK1 Q13546 2/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
TSHR P16473 1/20 0.38
SIGMAR1 Q99720 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9162328 0.79 CYP2C19 (0.39) CHRNB2CHRNB4CHRNA3CHRNA7CHRNA4
Hydrochloric Acid SCHEMBL9025807 0.74 TACR1 (0.44) CHRNB2CHRNB4CHRNA3CHRNA7CHRNA4
SCHEMBL4089851 0.72 TACR1 (0.55) SMN1; SMN2TSHR
SCHEMBL7255771 0.72 HRH3 (0.39) NPC1RAB9ASIGMAR1
SCHEMBL22462953 0.71 NPC1 (0.35) NPC1RAB9ASMN1; SMN2TSHR
SCHEMBL28710267 0.70 HRH3 (0.46) NPC1RAB9ASIGMAR1
SCHEMBL27908231 0.70 CHRNB2 (0.49) CHRNB2CHRNB4CHRNA3CHRNA7CHRNA4
SCHEMBL24697142 0.69 GBA1 (0.49) SIGMAR1
SCHEMBL22462978 0.69 BCHE (0.33) NPC1RAB9ASMN1; SMN2
SCHEMBL7101424 0.69 SPHK2 (0.40) CHRNB2CHRNA7CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2800738-B1 HETEROCYCLIC COMPOUNDS AND METHODS FOR THEIR USE NOVARTIS AG (CH) 2020-04-08 EP disclosed