SCHEMBL2184348

SCHEMBL2184348

CS(=O)(=O)c1ccc(N2CCC(O)CC2)c(F)c1

nearest known ligand 0.56

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 15/20 0.56
KCNH2 Q12809 2/20 0.47
AOC3 Q16853 1/20 0.45
GPR55 Q9Y2T6 1/20 0.45
GPR119 Q8TDV5 1/20 0.45
GAA P10253 1/20 0.44
ALDH1A1 P00352 1/20 0.44
LMNA P02545 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2937751 0.92 SLC6A9 (0.51) SLC6A9KCNH2GPR55GPR119
SCHEMBL2937750 0.92 SLC6A9 (0.51) SLC6A9KCNH2GPR55GPR119
SCHEMBL2939303 0.80 NOTUM (0.60) SLC6A9
SCHEMBL2937874 0.80 SLC6A9 (0.48) SLC6A9KCNH2GPR119
SCHEMBL2937875 0.80 SLC6A9 (0.48) SLC6A9KCNH2GPR119
SCHEMBL2939305 0.80 NOTUM (0.60) SLC6A9
SCHEMBL2182101 0.79 ALDH1A1 (0.57) SLC6A9KCNH2AOC3GPR55ALDH1A1
SCHEMBL2573793 0.79 SLC6A9 (0.55) SLC6A9KCNH2GPR55GAAALDH1A1
SCHEMBL12560142 0.79 SLC6A9 (0.62) SLC6A9ALDH1A1LMNA
SCHEMBL2937599 0.79 SLC6A9 (0.50) SLC6A9KCNH2AOC3GPR55GPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8293729-B2 Compounds, pharmaceutical composition and methods relating thereto BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-10-23 US disclosed
EP-2445878-A1 NEW COMPOUNDS, PHARMACEUTICAL COMPOSITION AND METHODS RELATING THERETO Boehringer Ingelheim International GmbH (DE) 2012-05-02 EP disclosed
US-20110166116-A1 NEW COMPOUNDS, PHARMACEUTICAL COMPOSITION AND METHODS RELATING THERETO BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-07-07 US disclosed
WO-2010149684-A1 NEW COMPOUNDS, PHARMACEUTICAL COMPOSITION AND METHODS RELATING THERETO BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-12-29 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110166116-A1 NEW COMPOUNDS, PHARMACEUTICAL COMPOSITION AND METHODS RELATING THERETO MC2R, REN, CYP11B2 SLC6A9 2874/4885KCNH2 2188/4885AOC3 2180/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.