SCHEMBL2186715

SCHEMBL2186715

O=C(O)c1ccsc1C(=O)Nc1ccccc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 2/20 0.63
ALDH1A1 P00352 2/20 0.58
HPGD P15428 5/20 0.57
KDM4E B2RXH2 2/20 0.57
GAA P10253 2/20 0.57
GLA P06280 1/20 0.57
MAPK1 P28482 1/20 0.57
CYP3A4 P08684 1/20 0.53
CYP2C9 P11712 1/20 0.53
ALOX12 P18054 1/20 0.53
PKM P14618 2/20 0.53
RXFP1 Q9HBX9 2/20 0.50
NPSR1 Q6W5P4 2/20 0.50
PRNP P04156 1/20 0.50
PPARG P37231 1/20 0.50
NCOR2 Q9Y618 1/20 0.50
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
LMNA P02545 2/20 0.47
TP53 P04637 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1124226 0.91 DHODH (0.78) DHODHALDH1A1HPGDKDM4EGAA
SCHEMBL2186276 0.86 DHODH (0.82) DHODHALDH1A1HPGDKDM4ECYP3A4
SCHEMBL2186832 0.85 RAB9A (0.58) DHODHALDH1A1HPGDKDM4EGAA
SCHEMBL2211815 0.80 KMT2A (0.58) GAARXFP1MEN1KMT2ALMNA
SCHEMBL1703428 0.79 DHODH (0.51) DHODHHPGDGAAPKMRXFP1
SCHEMBL1389175 0.79 PKM (0.74) ALDH1A1HPGDPKMPPARGNCOR2
SCHEMBL3640599 0.79 DHODH (0.51) DHODHALDH1A1HPGDKDM4EGAA
SCHEMBL1704235 0.78 LMNA (0.54) DHODHHPGDKDM4EPKMRXFP1
SCHEMBL11596321 0.78 RXFP1 (0.72) DHODHALDH1A1HPGDGAAPKM
SCHEMBL1810535 0.78 DHODH (1.00) DHODHALDH1A1HPGDKDM4EPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1578741-B1 AROMATIC COMPOUNDS AS ANTI-INFLAMMATORY, IMMUNOMODULATORY AND ANTI-PROLIFERATORY AGENTS 4SC AG (DE) 2011-07-13 EP claimed
EP-1578741-B1 AROMATIC COMPOUNDS AS ANTI-INFLAMMATORY, IMMUNOMODULATORY AND ANTI-PROLIFERATORY AGENTS 4SC AG (DE) 2011-07-13 EP disclosed