SCHEMBL21884555

SCHEMBL21884555

NC1NC1NC(=O)c1c(O)ccc(Cl)c1-c1ccccc1

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.37
MDM2 Q00987 2/20 0.37
FABP4 P15090 5/20 0.36
FABP3 P05413 4/20 0.36
HTT P42858 1/20 0.35
FABP5 Q01469 1/20 0.34
THRA P10827 1/20 0.34
THRB P10828 1/20 0.34
MAP2 P11137 2/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
ESR2 Q92731 1/20 0.33
SMYD3 Q9H7B4 1/20 0.32
GAA P10253 1/20 0.32
PTGS1 P23219 1/20 0.31
PTGS2 P35354 1/20 0.31
PPIA P62937 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21884595 0.75 FABP4 (0.39) FABP4FABP3HTTFABP5THRA
SCHEMBL27588764 0.65 ESR2 (0.52) FABP4FABP3HTTFABP5THRA
SCHEMBL1022491 0.61 ALDH1A1 (0.54) FABP4FABP3HTTFABP5THRA
SCHEMBL7106911 0.60 ESR2 (0.50) HTTTHRATHRBKDM4EALDH1A1
SCHEMBL4253909 0.60 CA12 (0.54) FABP4FABP3HTTKDM4EALDH1A1
SCHEMBL27505789 0.60 ESR2 (0.50) HTTTHRATHRBALDH1A1ESR2
SCHEMBL28999631 0.59 ESR2 (0.48) HTTTHRATHRBKDM4EALDH1A1
SCHEMBL28992361 0.59 KMT2A (0.55) FABP4FABP3FABP5MAP2KDM4E
SCHEMBL9469504 0.59 ALDH1A1 (0.45) FABP4FABP3HTTFABP5THRA
SCHEMBL11775117 0.58 THRB (0.54) HTTTHRBKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020061473-A1 SMALL MOLECULES TARGETING MUTANT MAMMALIAN PROTEINS JNANA THERAPEUTICS, INC. (US) 2020-03-26 WO disclosed