SCHEMBL218851

SCHEMBL218851

CC(=O)Oc1cc(S(=O)(=O)Cl)c2ccc3c(S(=O)(=O)Cl)cc(S(=O)(=O)Cl)c4ccc1c2c43

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.39
KDM4E B2RXH2 4/20 0.36
ALDH1A1 P00352 3/20 0.36
TSHR P16473 3/20 0.36
GAA P10253 2/20 0.36
RAB9A P51151 1/20 0.36
KMT2A Q03164 2/20 0.35
POLB P06746 2/20 0.35
MAPT P10636 2/20 0.35
BLM P54132 2/20 0.35
TDP1 Q9NUW8 2/20 0.35
APEX1 P27695 1/20 0.35
RECQL P46063 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
TRPV4 Q9HBA0 1/20 0.35
CFD P00746 1/20 0.35
ABCB11 O95342 1/20 0.35
PKM P14618 1/20 0.34
PIM1 P11309 1/20 0.33
BACE1 P56817 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9614315 0.97 HTT (0.39) HTTKDM4EALDH1A1TSHRGAA
SCHEMBL19939980 0.94 HTT (0.35) HTTKDM4EALDH1A1TSHRGAA
SCHEMBL9962926 0.89 KMT2A (0.42) HTTKDM4EALDH1A1TSHRGAA
SCHEMBL13039218 0.88 HTT (0.32) HTTKDM4EALDH1A1TSHRKMT2A
SCHEMBL9962933 0.86 ITGA1 (0.37) HTTKDM4EALDH1A1TSHRGAA
SCHEMBL168580 0.86 HTT (0.40) HTTKDM4EALDH1A1TSHRGAA
SCHEMBL29948312 0.86 HTT (0.40) HTTKDM4EALDH1A1TSHRGAA
SCHEMBL9717015 0.86 KMT2A (0.34) HTTKDM4EALDH1A1GAAKMT2A
SCHEMBL9962934 0.85 KMT2A (0.37) KDM4EALDH1A1GAAKMT2APOLB
SCHEMBL4925230 0.85 TRPV4 (0.33) TRPV4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 149 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9694357-B1 Multi-acid polymers and methods of making the same NISSAN NORTH AMERICA, INC. (US) 2017-07-04 US claimed
US-8951503-B2 Optical determination of glucose utilizing boronic acid adducts THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2015-02-10 US claimed
US-20090148956-A1 OPTICAL DETERMINATION OF GLUCOSE UTILIZING BORONIC ACID ADDUCTS SINGARAM BAKTHAN 2009-06-11 US claimed
US-7470420-B2 Optical determination of glucose utilizing boronic acid adducts THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2008-12-30 US claimed
EP-0396732-A4 FLUORESCENT IMMUNOASSAYS AND FLUORESCENT COMPOUNDS AND TRACERS THEREFORE 1992-10-07 EP claimed
EP-0396732-A1 FLUORESCENT IMMUNOASSAYS AND FLUORESCENT COMPOUNDS AND TRACERS THEREFORE DOWBEN, Robert M. (US) 1990-11-14 EP claimed
WO-1990005916-A1 FLUORESCENT IMMUNOASSAYS AND FLUORESCENT COMPOUNDS AND TRACERS THEREFORE DOWBEN ROBERT M (US) 1990-05-31 WO claimed
WO-2025021994-A1 NEW PHOTOCLEAVABLE PYRANINE DERIVATIVES, THEIR METHOD OF PREPARATION AND THEIR USES PARIS SCIENCES ET LETTRES (FR) 2025-01-30 WO disclosed
EP-3606639-B1 METHOD AND SYSTEM FOR SEPARATING BIOMOLECULES FROM A MIXTURE CONTAINING SAME UNIV RAMOT (IL) 2024-12-25 EP disclosed
WO-2024101447-A1 DIAGNOSIS METHOD, DIAGNOSIS DEVICE, AND ANTIBODY REGENERATION METHOD 国立大学法人信州大学 2024-05-16 WO disclosed
US-11673100-B2 Systems and methods for integrated solar photodialysis THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2023-06-13 US disclosed
US-11673100-B2 Systems and methods for integrated solar photodialysis THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2023-06-13 US disclosed
EP-2545373-B1 MEASURING ANALYTE CONCENTRATION INCORPORATING TEMPERATURE AND PH CORRECTION MEDTRONIC MINIMED INC (US) 2022-08-24 EP disclosed
EP-0396732-A4 FLUORESCENT IMMUNOASSAYS AND FLUORESCENT COMPOUNDS AND TRACERS THEREFORE 1992-10-07 EP disclosed
US-5094819-A FLUORESCENCE-BASED OPTICAL SENSOR AND METHOD FOR DETECTION OF LIPID-SOLUBLE ANALYTES WASHINGTON RESEARCH FOUNDATION (US) 1992-03-10 US disclosed
WO-1991000510-A1 FLUORESCENCE-BASED OPTICAL SENSOR FOR DETECTION OF LIPID-SOLUBLE ANALYTES WASHINGTON TECHNOLOGY CENTER (US) 1991-01-10 WO disclosed
EP-0396732-A1 FLUORESCENT IMMUNOASSAYS AND FLUORESCENT COMPOUNDS AND TRACERS THEREFORE DOWBEN, Robert M. (US) 1990-11-14 EP disclosed
US-4965087-A Method of making a sensor element for fluorescence-optical measurements AVL AG (CH) 1990-10-23 US disclosed
WO-1990005916-A1 FLUORESCENT IMMUNOASSAYS AND FLUORESCENT COMPOUNDS AND TRACERS THEREFORE DOWBEN ROBERT M (US) 1990-05-31 WO disclosed
US-4568518-A Sensor element for fluorescence-optical measurement AVL AG (CH) 1986-02-04 US disclosed