SCHEMBL21887773

SCHEMBL21887773

CC1Cn2nc(C(F)(F)F)cc2-c2ccc(Br)cc21

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 5/20 0.34
PTGS1 P23219 4/20 0.34
PDE4B Q07343 2/20 0.33
PDE3A Q14432 2/20 0.33
KDM1A O60341 2/20 0.31
HTR2A P28223 1/20 0.31
HTR2C P28335 1/20 0.31
HTR2B P41595 1/20 0.31
NT5E P21589 1/20 0.31
OPRM1 P35372 1/20 0.30
OPRD1 P41143 1/20 0.30
OPRK1 P41145 1/20 0.30
SLC6A4 P31645 1/20 0.30
HDAC3 O15379 1/20 0.30
HDAC4 P56524 1/20 0.30
HDAC1 Q13547 1/20 0.30
HDAC7 Q8WUI4 1/20 0.30
HDAC2 Q92769 1/20 0.30
HDAC10 Q969S8 1/20 0.30
HDAC11 Q96DB2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21888596 0.86 HTR2A (0.30) HTR2AHTR2CHTR2B
SCHEMBL21887738 0.79 HTR2A (0.32) HTR2AHTR2CHTR2BOPRM1OPRD1
SCHEMBL21888597 0.77 HTR2A (0.31) HTR2AHTR2CHTR2BSLC6A4
SCHEMBL21887870 0.71 ALDH1A1 (0.41)
SCHEMBL30875210 0.67 CTSK (0.32)
SCHEMBL24860256 0.64 PTGS1 (0.32) PTGS2PTGS1HDAC3HDAC4HDAC1
SCHEMBL30413203 0.64 PDK2 (0.38)
SCHEMBL30413996 0.64 PDK2 (0.38)
SCHEMBL31351756 0.63 MEN1 (0.43) HTR2AHTR2CHTR2BSLC6A4
SCHEMBL24934670 0.63 PTGS1 (0.31) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3626712-A2 LIVER X RECEPTOR (LXR) MODULATORS Ellora Therapeutics, Inc. (US) 2020-03-25 EP disclosed