SCHEMBL21887870

SCHEMBL21887870

CCOC(=O)c1cc2n(n1)CC(C)c1cc(Br)ccc1-2

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
TDP2 O95551 1/20 0.39
KMT2A Q03164 1/20 0.39
GABRG2 P18507 3/20 0.38
GABRB3 P28472 3/20 0.38
GABRA5 P31644 3/20 0.38
MAPT P10636 1/20 0.38
FAAH O00519 2/20 0.37
ELANE P08246 1/20 0.37
APAF1 O14727 1/20 0.37
SMAD3 P84022 1/20 0.37
KDM4E B2RXH2 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21888597 0.80 HTR2A (0.31)
SCHEMBL21887769 0.77 NR1H2 (0.59) FAAH
SCHEMBL21887738 0.73 HTR2A (0.32)
SCHEMBL15868151 0.72 SMN1; SMN2 (0.45) ALDH1A1SMN1; SMN2KMT2AGABRG2GABRB3
SCHEMBL21888596 0.72 HTR2A (0.30)
SCHEMBL21887773 0.71 PTGS2 (0.34)
SCHEMBL21607874 0.70 FAAH (0.45) ALDH1A1SMN1; SMN2KMT2AGABRG2GABRB3
SCHEMBL15868122 0.70 SMN1; SMN2 (0.45) ALDH1A1SMN1; SMN2GABRG2GABRB3GABRA5
SCHEMBL24456863 0.70 CYP1A2 (0.47) ALDH1A1TDP2KMT2AMAPT
SCHEMBL21598388 0.70 MARS1 (0.47) ALDH1A1SMN1; SMN2KMT2AFAAHELANE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3626712-A2 LIVER X RECEPTOR (LXR) MODULATORS Ellora Therapeutics, Inc. (US) 2020-03-25 EP disclosed