SCHEMBL21887738

SCHEMBL21887738

CC(C)c1cc2n(n1)CC(C)c1cc(Br)ccc1-2

nearest known ligand 0.32

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.32
HTR2C P28335 1/20 0.32
HTR2B P41595 1/20 0.32
OPRM1 P35372 1/20 0.32
OPRD1 P41143 1/20 0.32
OPRK1 P41145 1/20 0.32
SLC6A2 P23975 1/20 0.31
SLC6A4 P31645 1/20 0.31
SLC6A3 Q01959 1/20 0.31
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21888597 0.79 HTR2A (0.31) HTR2AHTR2CHTR2BSLC6A2SLC6A4
SCHEMBL21887773 0.79 PTGS2 (0.34) HTR2AHTR2CHTR2BOPRM1OPRD1
SCHEMBL21888596 0.78 HTR2A (0.30) HTR2AHTR2CHTR2B
SCHEMBL21887739 0.74 NR1H2 (0.53)
SCHEMBL21887870 0.73 ALDH1A1 (0.41)
SCHEMBL31351756 0.65 MEN1 (0.43) HTR2AHTR2CHTR2BSLC6A2SLC6A4
SCHEMBL24185333 0.64 GABRG2 (0.44) HTR2AHTR2CHTR2BOPRM1OPRD1
SCHEMBL4419838 0.63 PBRM1 (0.50) HTR2AHTR2CHTR2BOPRM1OPRD1
SCHEMBL31426351 0.61 HTR2B (0.38) HTR2AHTR2CHTR2BOPRM1OPRD1
SCHEMBL13437405 0.60 HTR2B (0.40) HTR2AHTR2CHTR2BOPRM1OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3626712-A2 LIVER X RECEPTOR (LXR) MODULATORS Ellora Therapeutics, Inc. (US) 2020-03-25 EP disclosed