SCHEMBL21895986

SCHEMBL21895986

C=C(c1ccccc1)[C@@]1(NC)CC1=O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.34
SMN1; SMN2 Q16637 4/20 0.34
MAPT P10636 4/20 0.34
LMNA P02545 3/20 0.34
XBP1 P17861 1/20 0.34
ATM Q13315 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
HPGD P15428 2/20 0.34
POLB P06746 1/20 0.33
ALDH1A1 P00352 3/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
DDB1 Q16531 1/20 0.33
CRBN Q96SW2 1/20 0.33
MEN1 O00255 4/20 0.32
KMT2A Q03164 4/20 0.32
CYP3A4 P08684 3/20 0.32
ALOX15 P16050 2/20 0.32
CES1 P23141 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9316282 0.65 ALDH1A1 (0.35) SMN1; SMN2MAPTLMNAXBP1ATM
SCHEMBL11495283 0.63 CES1 (0.42) TSHRSMN1; SMN2MAPTLMNAXBP1
Dimethylamine SCHEMBL607223 0.62 MEN1 (0.58) TSHRSMN1; SMN2MAPTLMNAXBP1
SCHEMBL7157657 0.62 KMT2A (0.43) TSHRSMN1; SMN2MAPTLMNAXBP1
Dimethylamine SCHEMBL8578211 0.61 CES1 (0.42) TSHRSMN1; SMN2MAPTLMNAXBP1
SCHEMBL4953900 0.61 MAOA (0.44) TSHRSMN1; SMN2MAPTLMNAXBP1
Dimethylamine SCHEMBL8980060 0.60 TSHR (0.46) TSHRSMN1; SMN2MAPTLMNAXBP1
SCHEMBL20630554 0.59 LMNA (0.42) SMN1; SMN2MAPTLMNAATMNPSR1
SCHEMBL21895900 0.59 LMNA (0.42) SMN1; SMN2MAPTLMNAATMNPSR1
Benzoic Acid SCHEMBL7547480 0.59 TSHR (0.70) TSHRSMN1; SMN2MAPTHPGDALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3636807-A1 CYCLIC PEPTIDE COMPOUND HAVING HIGH MEMBRANE PERMEABILITY, AND LIBRARY CONTAINING SAME Chugai Seiyaku Kabushiki Kaisha (JP) 2020-04-15 EP disclosed