SCHEMBL21899548

SCHEMBL21899548

N=C(Br)c1c(N)ncnc1NC1CCCN(C(=O)CCCl)C1

nearest known ligand 0.49

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
BTK Q06187 10/20 0.49
JAK3 P52333 9/20 0.42
PIK3CD O00329 1/20 0.42
PIK3R1 P27986 1/20 0.42
PIK3CA P42336 1/20 0.42
EGFR P00533 1/20 0.42
JAK1 P23458 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21900351 0.91 BTK (0.49) BTKJAK3PIK3CDEGFRJAK1
SCHEMBL21900774 0.90 BTK (0.51) BTKJAK3PIK3CDPIK3R1PIK3CA
SCHEMBL19649309 0.81 BTK (0.65) BTKEGFR
SCHEMBL14647420 0.80 BTK (0.50) BTKJAK3PIK3CDEGFRJAK1
SCHEMBL21899804 0.79 BTK (0.47) BTKJAK3EGFRJAK1
SCHEMBL21899550 0.78 BTK (0.44) BTKJAK3EGFRJAK1
SCHEMBL19623270 0.77 BTK (0.51) BTKJAK3PIK3CDPIK3R1PIK3CA
SCHEMBL24464321 0.75 HPGDS (0.44) EGFRJAK1
SCHEMBL18618516 0.73 BTK (0.67) BTKJAK3EGFRJAK1
SCHEMBL21899554 0.73 BTK (0.67) BTKJAK3EGFRJAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3257855-B1 METHOD FOR PREPARING IBRUTINIB SHANGHAI DUDE MEDICAL SCIENCE AND TECH CO LTD (CN) 2020-04-22 EP disclosed