SCHEMBL2191285

SCHEMBL2191285

Cn1cnc(-c2nc(N)c3ccc(C(F)(F)F)nc3n2)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 2/20 0.47
ADORA2A P29274 1/20 0.47
ALDH1A1 P00352 3/20 0.38
KDM4E B2RXH2 3/20 0.38
KMT2A Q03164 1/20 0.38
GAA P10253 2/20 0.37
ADORA3 P0DMS8 1/20 0.36
LRRK2 Q5S007 1/20 0.34
MAPT P10636 2/20 0.33
TEAD1 P28347 1/20 0.33
YAP1 P46937 1/20 0.33
RAB9A P51151 1/20 0.33
MAT2A P31153 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
RORC P51449 1/20 0.32
MDM2 Q00987 1/20 0.32
KCNH2 Q12809 1/20 0.31
EGFR P00533 1/20 0.31
FGFR1 P11362 1/20 0.31
KDR P35968 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2190316 0.76 ADORA1 (0.53) ADORA1ADORA2AADORA3LRRK2
SCHEMBL2188560 0.73 ADORA1 (0.58) ADORA1ADORA2AALDH1A1KDM4EGAA
SCHEMBL30500672 0.70 ALDH1A1 (0.45) ADORA1ALDH1A1KDM4EKMT2AGAA
SCHEMBL2186774 0.69 ADORA2A (0.46) ADORA1ADORA2AADORA3LRRK2MAPT
SCHEMBL2187983 0.69 ADORA2A (0.56) ADORA1ADORA2ALRRK2FGFR1KDR
SCHEMBL2184224 0.69 ADORA2A (0.47) ADORA1ADORA2ALRRK2FGFR1KDR
SCHEMBL2185605 0.68 ADORA2A (0.46) ADORA1ADORA2ALRRK2MAPT
SCHEMBL30500674 0.67 ALDH1A1 (0.42) ADORA1ALDH1A1KDM4EKMT2AGAA
SCHEMBL13853257 0.66 ADK (0.44) ALDH1A1KDM4EKMT2AGAALRRK2
SCHEMBL2244688 0.65 PAK4 (0.41) ALDH1A1GAAMAPTRAB9AMAT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346859-A1 HETEROCYCLIC JAK KINASE INHIBITORS AstraZeneca AB (SE) 2011-07-27 EP disclosed