SCHEMBL21921827

SCHEMBL21921827

NCc1ccc(OCCC(F)(F)F)cn1

nearest known ligand 0.36

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.36
MCHR1 Q99705 1/20 0.36
MAOB P27338 2/20 0.36
LTA4H P09960 1/20 0.34
HTR2A P28223 3/20 0.34
KEAP1 Q14145 1/20 0.33
NFE2L2 Q16236 1/20 0.33
ACACB O00763 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5728790 0.87 HRH3 (0.35) HRH3LTA4H
SCHEMBL507036 0.83 ALDH1A1 (0.43) MAOB
SCHEMBL22604312 0.79 NCF1 (0.41) HRH3LTA4H
SCHEMBL15901127 0.76 CHRNB2 (0.39) MCHR1MAOBACACB
SCHEMBL11411633 0.74 MAOB (0.40) HRH3MAOB
Hydrochloric Acid SCHEMBL13736278 0.74 LNPEP (0.43) MCHR1MAOBHTR2A
SCHEMBL16853366 0.74 ST14 (0.40) HRH3LTA4H
SCHEMBL507305 0.72 MBOAT4 (0.37) MAOB
SCHEMBL15350553 0.71 P4HTM (0.55) ACACB
SCHEMBL507873 0.71 MBOAT4 (0.34) ACACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3632899-A1 ARYL SUBSTITUTED CARBOXAMIDE DERIVATIVES AS CALCIUM OR SODIUM CHANNEL BLOCKERS RaQualia Pharma Inc. (JP) 2020-04-08 EP disclosed