SCHEMBL21923049

SCHEMBL21923049

Ic1ccc(-n2cnnc2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.52
CYP2C9 P11712 2/20 0.52
QPCT Q16769 1/20 0.45
FAAH O00519 1/20 0.39
MGLL Q99685 1/20 0.39
LMNA P02545 2/20 0.37
RXFP1 Q9HBX9 1/20 0.37
KMT2A Q03164 2/20 0.36
HDAC8 Q9BY41 1/20 0.33
ADH5 P11766 1/20 0.33
CA12 O43570 1/20 0.33
CA9 Q16790 1/20 0.33
ABL1 P00519 1/20 0.32
SRC P12931 1/20 0.32
MAPT P10636 1/20 0.31
ENPP2 Q13822 1/20 0.31
MKNK1 Q9BUB5 1/20 0.31
MKNK2 Q9HBH9 1/20 0.31
NOTUM Q6P988 1/20 0.31
MPO P05164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12841347 0.74 CYP1A2 (0.52) CYP1A2CYP2C9QPCTMGLLLMNA
SCHEMBL1352015 0.74 MAPT (0.56) CYP1A2CYP2C9QPCTLMNARXFP1
SCHEMBL17690362 0.74 CYP1A2 (0.52) CYP1A2CYP2C9QPCTLMNARXFP1
SCHEMBL6518759 0.74 CYP2C9 (0.58) CYP1A2CYP2C9QPCTMGLLLMNA
SCHEMBL1186988 0.74 ENPP2 (0.56) CYP1A2CYP2C9QPCTMGLLLMNA
SCHEMBL256624 0.72 CYP3A4 (0.52) CYP1A2CYP2C9QPCTLMNAKMT2A
SCHEMBL31387623 0.72 CYP1A2 (0.50) CYP1A2CYP2C9QPCTLMNARXFP1
SCHEMBL17672944 0.72 LMNA (0.64) CYP1A2CYP2C9LMNAKMT2AADH5
SCHEMBL393880 0.70 KDM4E (0.50) CYP1A2FAAHMGLLKMT2AMAPT
SCHEMBL2511973 0.70 KCNJ1 (0.53) CYP1A2CYP2C9QPCTRXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3169673-B1 INHIBITORS OF THE RENAL OUTER MEDULLARY POTASSIUM CHANNEL MERCK SHARP & DOHME (US) 2020-04-29 EP disclosed