SCHEMBL21940467

SCHEMBL21940467

Nc1cc(OCC2CC2(F)F)nc(C(F)(F)F)c1

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 3/20 0.36
HSP90AA1 P07900 1/20 0.34
HSP90AB1 P08238 1/20 0.34
LOXL2 Q9Y4K0 4/20 0.33
FFAR2 O15552 1/20 0.32
MBOAT4 Q96T53 2/20 0.32
APP P05067 1/20 0.32
BACE1 P56817 1/20 0.32
ALDH1A1 P00352 1/20 0.32
MAPT P10636 1/20 0.32
RORC P51449 1/20 0.31
SCN8A Q9UQD0 1/20 0.31
SCN10A Q9Y5Y9 1/20 0.31
ACACB O00763 4/20 0.31
KDM4E B2RXH2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21940590 0.85 IDH1 (0.37) IDH1HSP90AA1HSP90AB1LOXL2FFAR2
SCHEMBL20606883 0.76 HSP90AA1 (0.42) HSP90AA1HSP90AB1LOXL2ALDH1A1MAPT
SCHEMBL20606969 0.75 CA2 (0.39) LOXL2
SCHEMBL21940313 0.74 MCHR1 (0.43) LOXL2SCN8A
SCHEMBL21940469 0.73 HSP90AA1 (0.35) HSP90AA1HSP90AB1LOXL2MBOAT4ALDH1A1
SCHEMBL21940793 0.73 NUDT1 (0.41) HSP90AA1HSP90AB1LOXL2ALDH1A1MAPT
SCHEMBL21940508 0.73 GPR84 (0.41)
SCHEMBL21941067 0.72 TLR7 (0.39) HSP90AA1HSP90AB1LOXL2ALDH1A1MAPT
SCHEMBL20606902 0.72 HSP90AA1 (0.39) HSP90AA1HSP90AB1LOXL2ALDH1A1MAPT
SCHEMBL20606989 0.71 HSP90AA1 (0.38) HSP90AA1HSP90AB1LOXL2ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3423445-B1 NOVEL COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS THEREOF FOR THE TREATMENT OF FIBROSIS GALAPAGOS NV (BE) 2020-04-01 EP disclosed