SCHEMBL21940807

SCHEMBL21940807

Cc1cc(CN)nnc1N1CCOC(CN(C)C)C1

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 7/20 0.44
ADORA2A P29274 1/20 0.39
ADORA1 P30542 1/20 0.39
CHEK1 O14757 9/20 0.38
CHEK2 O96017 8/20 0.34
AOC3 Q16853 1/20 0.34
PTPN11 Q06124 1/20 0.34
SYK P43405 1/20 0.32
STK3 Q13188 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21940810 0.82 LRRK2 (0.41) LRRK2ADORA2AADORA1CHEK1AOC3
SCHEMBL21941085 0.80 LRRK2 (0.50) LRRK2ADORA2AADORA1CHEK1CHEK2
SCHEMBL21940805 0.79 ELOVL1 (0.39)
SCHEMBL17623325 0.72 LRRK2 (0.48) LRRK2CHEK1CHEK2
SCHEMBL21940286 0.71 ALDH1A1 (0.42) ADORA2AADORA1
SCHEMBL21262293 0.70 GRIN2D (0.43) LRRK2ADORA2AADORA1CHEK1CHEK2
SCHEMBL21940600 0.69 LRRK2 (0.41) LRRK2ADORA2AADORA1STK3
SCHEMBL16440191 0.69 GAA (0.43) LRRK2SYK
SCHEMBL31200599 0.69 ADORA2A (0.50) LRRK2ADORA2AADORA1AOC3PTPN11
SCHEMBL21941081 0.68 AKT1 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3423445-B1 NOVEL COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS THEREOF FOR THE TREATMENT OF FIBROSIS GALAPAGOS NV (BE) 2020-04-01 EP disclosed