SCHEMBL2197181

SCHEMBL2197181

CC(C)(C)c1ccc(Nc2ccc(-c3ccc4c(c3)C(=O)N(C3(OC=O)CCCC3)C4)cc2)cc1

nearest known ligand 0.33

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
OPRD1 P41143 1/20 0.31
MAP3K5 Q99683 1/20 0.31
XDH P47989 1/20 0.31
SLC22A12 Q96S37 1/20 0.31
HRH3 Q9Y5N1 1/20 0.31
KIF11 P52732 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2184971 0.89 MEN1 (0.41) HDAC6
SCHEMBL2202235 0.87 JAK2 (0.38)
SCHEMBL2194266 0.87 APP (0.36)
SCHEMBL2196756 0.85 JAK2 (0.38)
SCHEMBL2198728 0.83 JAK2 (0.39)
SCHEMBL2199101 0.82 ALDH1A1 (0.37) HRH3
SCHEMBL2197176 0.81 KIF11 (0.38) HDAC4HDAC1HDAC6MAP3K5XDH
SCHEMBL2179546 0.77 NPC1 (0.42)
SCHEMBL2179901 0.77 SLC2A1 (0.42) XDH
SCHEMBL13718920 0.76 TRPV1 (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2519500-A1 INHIBITORS OF DIACYLGLYCEROL ACYL TRANSFERASE Piramal Healthcare Ltd. (IN) 2012-11-07 EP disclosed
WO-2011080718-A1 INHIBITORS OF DIACYLGLYCEROL ACYL TRANSFERASE PIRAMAL LIFE SCIENCES LIMITED (IN) 2011-07-07 WO disclosed