SCHEMBL22007454

SCHEMBL22007454

CC(C)(C)c1ccc(-c2c3ccccc3c(-c3ccc4oc5cc(-c6cccc7ccccc67)ccc5c4c3)c3ccccc23)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR84 Q9NQS5 1/20 0.38
ALDH1A1 P00352 1/20 0.37
MAPT P10636 1/20 0.37
HSP90AA1 P07900 1/20 0.36
HSP90AB1 P08238 1/20 0.36
PPARG P37231 2/20 0.34
PPARA Q07869 2/20 0.34
PSD A5PKW4 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
PPARD Q03181 1/20 0.34
MAOA P21397 1/20 0.34
MAOB P27338 1/20 0.34
MCL1 Q07820 1/20 0.33
ACMSD Q8TDX5 1/20 0.33
ENPP3 O14638 1/20 0.33
ENPP1 P22413 1/20 0.33
CCR4 P51679 1/20 0.33
MAP1LC3B Q9GZQ8 1/20 0.33
MAP1LC3A Q9H492 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9890831 0.95 GPR84 (0.41) GPR84ALDH1A1MAPTPPARGPPARA
SCHEMBL22947726 0.88 MCL1 (0.40) ALDH1A1MAPTHSP90AA1HSP90AB1PSD
SCHEMBL23437638 0.87 MCL1 (0.39) ALDH1A1MAPTHSP90AA1HSP90AB1PSD
SCHEMBL24982657 0.87 PSD (0.39) ALDH1A1MAPTHSP90AA1HSP90AB1PSD
SCHEMBL25624553 0.87 ALOX5 (0.41) ALDH1A1MAPTHSP90AA1HSP90AB1PSD
SCHEMBL23427150 0.86 CA12 (0.39) ALDH1A1MAPTMCL1ACMSDENPP3
SCHEMBL23427461 0.86 CA12 (0.39) ALDH1A1MAPTMCL1ACMSDENPP3
SCHEMBL27372132 0.85 ALOX5 (0.38) ALDH1A1MAPTHSP90AA1HSP90AB1PSD
SCHEMBL24173562 0.84 ALOX5 (0.41) ALDH1A1MAPTHSP90AA1HSP90AB1CYP2C19
SCHEMBL23814473 0.84 ALOX5 (0.41) GPR84ALDH1A1MAPTHSP90AA1HSP90AB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 34 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12030900-B2 Boron compound and organic light-emitting diode comprising same SFC CO., LTD. (KR) 2024-07-09 US disclosed
US-12018039-B2 Boron compound, and organic light-emitting diode comprising same SFC CO., LTD. (KR) 2024-06-25 US disclosed
US-12018039-B2 Boron compound, and organic light-emitting diode comprising same SFC CO., LTD. (KR) 2024-06-25 US disclosed
US-20240018164-A1 POLYCYCLIC AROMATIC DERIVATIVE COMPOUND AND ORGANOELECTROLUMINESCENT DEVICE USING SAME SFC CO., LTD. (KR) 2024-01-18 US disclosed
US-20240018164-A1 POLYCYCLIC AROMATIC DERIVATIVE COMPOUND AND ORGANOELECTROLUMINESCENT DEVICE USING SAME SFC CO., LTD. (KR) 2024-01-18 US disclosed
EP-3889236-B1 ORGANIC LIGHT-EMITTING ELEMENT USING POLYCYCLIC AROMATIC DERIVATIVE COMPOUND SFC CO LTD (KR) 2023-11-22 EP disclosed
US-20230329109-A1 POLYCYCLIC AROMATIC DERIVATIVE COMPOUND AND ORGANOELECTROLUMINESCENT DEVICE USING SAME SFC CO., LTD. (KR) 2023-10-12 US disclosed
US-20230329109-A1 POLYCYCLIC AROMATIC DERIVATIVE COMPOUND AND ORGANOELECTROLUMINESCENT DEVICE USING SAME SFC CO., LTD. (KR) 2023-10-12 US disclosed
US-20230287010-A1 POLYCYCLIC AROMATIC DERIVATIVE COMPOUND AND ORGANIC LIGHT-EMITTING DEVICE USING SAME SFC CO., LTD (KR) 2023-09-14 US disclosed
US-20230287010-A1 POLYCYCLIC AROMATIC DERIVATIVE COMPOUND AND ORGANIC LIGHT-EMITTING DEVICE USING SAME SFC CO., LTD (KR) 2023-09-14 US disclosed
US-20210403490-A1 NOVEL BORON COMPOUND, AND ORGANIC LIGHT-EMITTING DIODE COMPRISING SAME SFC CO., LTD. (KR) 2021-12-30 US disclosed
US-20210317144-A1 Boron compound and organic light emitting diode including the same SFC CO., LTD. (KR) 2021-10-14 US disclosed
US-20210305514-A1 POLYCYCLIC AROMATIC COMPOUND AND ORGANOELECTROLUMINESCENT DEVICE USING THE SAME SFC CO., LTD. (KR) 2021-09-30 US disclosed
US-20210167293-A1 POLYCYCLIC AROMATIC COMPOUNDS AND ORGANIC ELECTROLUMINESCENT DEVICES USING THE SAME SFC CO., LTD. (KR) 2021-06-03 US disclosed
EP-3660024-B1 POLYCYCLIC AROMATIC COMPOUNDS AND ORGANIC ELECTROLUMINESCENT DEVICES USING THE SAME SFC CO LTD (KR) 2021-05-05 EP disclosed
US-10981938-B2 Polycyclic aromatic compounds and organic electroluminescent devices using the same SFC CO., LTD. (KR) 2021-04-20 US disclosed
US-20200395553-A1 ORGANIC ELECTROLUMINESCENT DEVICE SFC CO., LTD. (KR) 2020-12-17 US disclosed
US-20200172558-A1 POLYCYCLIC AROMATIC COMPOUNDS AND ORGANIC ELECTROLUMINESCENT DEVICES USING THE SAME SFC CO., LTD. (KR) 2020-06-04 US disclosed
EP-3660024-A1 POLYCYCLIC AROMATIC COMPOUNDS AND ORGANIC ELECTROLUMINESCENT DEVICES USING THE SAME SFC Co., Ltd. (KR) 2020-06-03 EP disclosed
US-20200161552-A1 INDOLOCARBAZOLE DERIVATIVES AND ORGANIC ELECTROLUMINESCENT DEVICES USING THE SAME SFC CO., LTD. (KR) 2020-05-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (12 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210317144-A1 Boron compound and organic light emitting diode including the same CLTB, CD79B, BLVRB GPR84 2107/4885ALDH1A1 102/4885MAPT 932/4885
US-20230287010-A1 POLYCYCLIC AROMATIC DERIVATIVE COMPOUND AND ORGANIC LIGHT-EMITTING DEVICE USING SAME DDT, TYR, DDC GPR84 1665/4885ALDH1A1 608/4885MAPT 219/4885
US-20200172558-A1 POLYCYCLIC AROMATIC COMPOUNDS AND ORGANIC ELECTROLUMINESCENT DEVICES USING THE SAME DDC, TYR, DDT GPR84 3319/4885ALDH1A1 711/4885MAPT 1909/4885
US-20210403490-A1 NOVEL BORON COMPOUND, AND ORGANIC LIGHT-EMITTING DIODE COMPRISING SAME CLTB, CD79B, CYBA GPR84 1996/4885ALDH1A1 113/4885MAPT 970/4885
US-12018039-B2 Boron compound, and organic light-emitting diode comprising same CLTB, CD79B, CYBA GPR84 2558/4885ALDH1A1 103/4885MAPT 1036/4885
US-20240018164-A1 POLYCYCLIC AROMATIC DERIVATIVE COMPOUND AND ORGANOELECTROLUMINESCENT DEVICE USING SAME DDT, UROD, DDC GPR84 1041/4885ALDH1A1 307/4885MAPT 1629/4885
US-20210167293-A1 POLYCYCLIC AROMATIC COMPOUNDS AND ORGANIC ELECTROLUMINESCENT DEVICES USING THE SAME DDC, TYR, DDT GPR84 3319/4885ALDH1A1 711/4885MAPT 1909/4885
US-20230329109-A1 POLYCYCLIC AROMATIC DERIVATIVE COMPOUND AND ORGANOELECTROLUMINESCENT DEVICE USING SAME DDT, UROD, DDC GPR84 816/4885ALDH1A1 269/4885MAPT 1234/4885
US-10981938-B2 Polycyclic aromatic compounds and organic electroluminescent devices using the same DDC, TYR, DDT GPR84 3319/4885ALDH1A1 711/4885MAPT 1909/4885
US-12030900-B2 Boron compound and organic light-emitting diode comprising same CLTB, CD79B, CYBA GPR84 2577/4885ALDH1A1 170/4885MAPT 950/4885
US-20200395553-A1 ORGANIC ELECTROLUMINESCENT DEVICE LEF1, AP2A2, CCNA1 GPR84 3706/4885ALDH1A1 17/4885MAPT 2312/4885
US-20210305514-A1 POLYCYCLIC AROMATIC COMPOUND AND ORGANOELECTROLUMINESCENT DEVICE USING THE SAME TYR, DDC, PAH GPR84 2264/4885ALDH1A1 733/4885MAPT 3753/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.