SCHEMBL22010534

SCHEMBL22010534

COc1ccc(CN(C)Cc2c(C)sc3c(O)cccc23)cc1

nearest known ligand 0.57

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.57
MEN1 O00255 3/20 0.57
ACHE P22303 3/20 0.44
SMPD1 P17405 1/20 0.40
PYCR1 P32322 1/20 0.40
TDP1 Q9NUW8 1/20 0.39
TSHR P16473 1/20 0.38
ACKR3 P25106 1/20 0.37
GNRHR P30968 2/20 0.37
ALOX5 P09917 1/20 0.37
BCHE P06276 2/20 0.36
POLB P06746 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21963819 0.86 KMT2A (0.48) KMT2AMEN1ACHESMPD1PYCR1
SCHEMBL22010529 0.81 KMT2A (0.44) KMT2AMEN1ACHESMPD1PYCR1
SCHEMBL31033278 0.81 KMT2A (0.44) KMT2AMEN1ACHESMPD1PYCR1
SCHEMBL21964039 0.76 KMT2A (0.57) KMT2AMEN1ACHESMPD1PYCR1
SCHEMBL4611890 0.71 PYCR1 (0.69) KMT2AMEN1ACHESMPD1PYCR1
SCHEMBL16039094 0.68 ACHE (0.76) KMT2AMEN1ACHESMPD1PYCR1
SCHEMBL22010475 0.67 KMT2A (0.48) KMT2AMEN1ACHESMPD1PYCR1
SCHEMBL9821873 0.66 CYP2D6 (0.68) KMT2AMEN1ACHESMPD1TDP1
SCHEMBL20804510 0.66 PYCR1 (0.62) KMT2AMEN1ACHESMPD1PYCR1
SCHEMBL9416597 0.66 ACHE (0.59) KMT2AMEN1ACHEPYCR1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113272302-A Antibiotic compounds, process for their manufacture, pharmaceutical compositions containing them and their use 德彪药业国际股份公司 2021-08-17 CN disclosed
WO-2020099341-A1 ANTIBIOTIC COMPOUNDS, METHODS OF MANUFACTURING THE SAME, PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME AND USES THEREOF DEBIOPHARM INTERNATIONAL S.A. (CH) 2020-05-22 WO disclosed