SCHEMBL22044273

SCHEMBL22044273

N/C=N\N=C(/N)c1ccc(F)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 5/20 0.44
GRIN2D O15399 4/20 0.44
GRIN3B O60391 4/20 0.44
GRIN1 Q05586 4/20 0.44
GRIN2A Q12879 4/20 0.44
GRIN2C Q14957 4/20 0.44
GRIN3A Q8TCU5 4/20 0.44
PAX8 Q06710 1/20 0.42
NPC1 O15118 3/20 0.41
RAB9A P51151 3/20 0.41
PKM P14618 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.40
SLC22A2 O15244 1/20 0.38
SLC22A1 O15245 1/20 0.38
SLC22A3 O75751 1/20 0.38
PLAU P00749 1/20 0.38
CES2 O00748 1/20 0.37
CES1 P23141 1/20 0.37
KMT2A Q03164 1/20 0.37
TAAR1 Q96RJ0 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23031878 0.86 LMNA (0.44) GRIN2BKMT2A
SCHEMBL23031877 0.83 PYCR1 (0.41) GRIN2BNPC1RAB9ASMN1; SMN2KMT2A
SCHEMBL22815269 0.82 KDM1A (0.48) NPC1RAB9APKMSMN1; SMN2KMT2A
SCHEMBL23032115 0.81 L3MBTL1 (0.58) SMN1; SMN2KMT2A
SCHEMBL22043779 0.80 CYP2D6 (0.47) GRIN2BGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL18891357 0.79 KMT2A (0.48) GRIN2BGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL22044405 0.78 PARP1 (0.50) GRIN2BNPC1RAB9APKMCES2
SCHEMBL21300883 0.77 LOXL2 (0.47) PLAUNOS3NOS1
SCHEMBL21889662 0.76 GRIN2D (0.49) GRIN2BGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL24022848 0.75 HDAC1 (0.50) GRIN2BGRIN2DGRIN3BGRIN1GRIN2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3909944-A1 NUCLIDE LABELLED H-TETRAZINES AND USE THEREOF FOR PET AND SPECT PRETARGETED IMAGING AND RADIONUCLIDE THERAPY Rigshospitalet (DK) 2021-11-17 EP disclosed
WO-2020108720-A1 NOVEL TETRAZINE COMPOUNDS FOR IN VIVO IMAGING Københavns Universitet (DK) 2020-06-04 WO disclosed