Enclomiphene

Enclomiphene

SCHEMBL220459

CCN(CC)CCOc1ccc(/C(=C(/Cl)c2ccccc2)c2ccccc2)cc1.O=C(O)CC(O)(CC(=O)O)C(=O)O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ESR1

The experimentally established mechanism targets of Enclomiphene. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 known ✓ P03372 10/20 0.75
KDM4E B2RXH2 6/20 1.00
KMT2A Q03164 5/20 1.00
CYP2D6 P10635 5/20 1.00
MEN1 O00255 4/20 1.00
LMNA P02545 4/20 1.00
CYP1A2 P05177 4/20 1.00
MAPT P10636 3/20 1.00
TP53 P04637 2/20 1.00
CYP2C9 P11712 2/20 1.00
MAPK1 P28482 2/20 1.00
EBP Q15125 5/20 0.75
SIGMAR1 Q99720 3/20 0.75
KCNH2 Q12809 2/20 0.75
CHRM2 P08172 2/20 0.75
ADRA2A P08913 2/20 0.75
ADORA3 P0DMS8 2/20 0.75
CHRM1 P11229 2/20 0.75
PTGS1 P23219 2/20 0.75
SLC6A2 P23975 2/20 0.75

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Enclomiphene SCHEMBL8040981 1.00 KDM4E (1.00) KDM4EKMT2ACYP2D6MEN1LMNA
Zuclomiphene SCHEMBL223472 1.00 KDM4E (1.00) KDM4EKMT2ACYP2D6MEN1LMNA
Clomiphene SCHEMBL220953 1.00 KDM4E (1.00) KDM4EKMT2ACYP2D6MEN1LMNA
Clomiphene SCHEMBL20942789 1.00 KDM4E (1.00) KDM4EKMT2ACYP2D6MEN1LMNA
Clomiphene SCHEMBL27599894 1.00 KDM4E (1.00) KDM4EKMT2ACYP2D6MEN1LMNA
Citric Acid SCHEMBL8616232 0.94 KMT2A (0.89) KDM4EKMT2ACYP2D6MEN1LMNA
Citric Acid SCHEMBL8614802 0.94 KMT2A (0.89) KDM4EKMT2ACYP2D6MEN1LMNA
Citric Acid SCHEMBL8614814 0.94 KMT2A (0.89) KDM4EKMT2ACYP2D6MEN1LMNA
Citric Acid SCHEMBL8612826 0.93 KMT2A (0.87) KDM4EKMT2ACYP2D6MEN1LMNA
Citric Acid SCHEMBL8613135 0.93 KMT2A (0.87) KDM4EKMT2ACYP2D6MEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1601 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12569624-B2 Devices, methods and compositions for reproductive organs FEMASYS INC. (US) 2026-03-10 US claimed
US-12544387-B2 Methods and compositions for testosterone production SEPAH SAVIZ CAMERON (US) 2026-02-10 US claimed
US-12533364-B2 Methods and compositions for testosterone production Saviz SEPAH (US) 2026-01-27 US claimed
US-12533363-B2 Methods and compositions for testosterone production Sepah, Saviz (US) 2026-01-27 US claimed
EP-4680248-A1 PRODUCTS OF MANUFACTURE AND THERAPEUTIC COMPOSITIONS FOR TREATING, AMELIORATING OR PREVENTING VIRAL INFECTIONS AND METHODS FOR MAKING AND USING THEM Topelia Aust Limited (ACN 652 771 670) (AU) 2026-01-21 EP claimed
US-20250295670-A1 METHODS AND COMPOSITIONS FOR TESTOSTERONE PRODUCTION SEPAH SAVIZ CAMERON (US) 2025-09-25 US claimed
US-20250288598-A1 METHODS AND COMPOSITIONS FOR TESTOSTERONE PRODUCTION Maximus Health, Inc. 2025-09-18 US claimed
US-20250281505-A1 METHODS AND COMPOSITIONS FOR TESTOSTERONE PRODUCTION Maximus Health, Inc. 2025-09-11 US claimed
US-20250269005-A1 METHODS FOR TREATING, AMELIORATING OR PREVENTING INFECTIONS USING DRUG AND VACCINATION COMBINATION TREATMENT TOPELIA AUST LIMITED (ACN 652 771 670) (AU) 2025-08-28 US claimed
US-20250268915-A1 METHODS AND COMPOSITIONS FOR TESTOSTERONE PRODUCTION Maximus Health, Inc. (US) 2025-08-28 US claimed
EP-1216024-A4 FORMULATION FOR MENOPAUSAL WOMEN DRUGTECH CORP (US) 2005-02-02 EP claimed
EP-1471917-A1 USE OF PDE5 INHIBITORS SUCH AS SILDENAFIL IN THE TREATMENT OF POLYCYSTIC OVARY SYNDROME Pfizer Limited (GB) 2004-11-03 EP claimed
US-20040029891-A1 Use of PDE5 inhibitors in the treatment of polycystic ovary syndrome PFIZER INC. 2004-02-12 US claimed
WO-2003066061-A1 USE OF PDE5 INHIBITORS SUCH AS SILDENAFIL IN THE TREATMENT OF POLYCYSTIC OVARY SYNDROME PFIZER LIMITED (GB) 2003-08-14 WO claimed
US-20020173510-A1 Formulation for menopausal women DRUGTECH CORPORATION 2002-11-21 US claimed
US-6479545-B1 Formulation for menopausal women DRUGTECH CORPORATION 2002-11-12 US claimed
US-20020137749-A1 Formulation for menopausal women DRUGTECH CORPORATION (US) 2002-09-26 US claimed
EP-1216024-A1 FORMULATION FOR MENOPAUSAL WOMEN Drugtech Corporation (US) 2002-06-26 EP claimed
WO-2001024772-A1 FORMULATION FOR MENOPAUSAL WOMEN DRUGTECH CORPORATION (US) 2001-04-12 WO claimed
WO-2000077590-A1 APPARATUS FOR CALCULATING TIME PERIODS AND FUTURE DATES CRAIG H RANDALL (US) 2000-12-21 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (12 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250268915-A1 METHODS AND COMPOSITIONS FOR TESTOSTERONE PRODUCTION SHBG, AR, CYP17A1 ESR1 15/4885KDM4E 3258/4885KMT2A 4203/4885
US-20250295670-A1 METHODS AND COMPOSITIONS FOR TESTOSTERONE PRODUCTION SHBG, AR, CYP17A1 ESR1 15/4885KDM4E 3258/4885KMT2A 4203/4885
US-12544387-B2 Methods and compositions for testosterone production SHBG, FSHR, GNRHR ESR1 27/4885KDM4E 3190/4885KMT2A 3116/4885
US-20250281505-A1 METHODS AND COMPOSITIONS FOR TESTOSTERONE PRODUCTION SHBG, AR, CYP19A1 ESR1 11/4885KDM4E 2748/4885KMT2A 3988/4885
US-20250288598-A1 METHODS AND COMPOSITIONS FOR TESTOSTERONE PRODUCTION SHBG, AR, CYP19A1 ESR1 11/4885KDM4E 2748/4885KMT2A 3988/4885
US-20250269005-A1 METHODS FOR TREATING, AMELIORATING OR PREVENTING INFECTIONS USING DRUG AND VACCINATION COMBINATION TREATMENT ZFX, ACE2, ZFR ESR1 1685/4885KDM4E 303/4885KMT2A 641/4885
US-20040029891-A1 Use of PDE5 inhibitors in the treatment of polycystic ovary syndrome PDE5A, PDE12, PDE2A ESR1 3837/4885KDM4E 1325/4885KMT2A 2350/4885
US-12533363-B2 Methods and compositions for testosterone production SHBG, FSHR, GNRHR ESR1 27/4885KDM4E 2780/4885KMT2A 3523/4885
US-12569624-B2 Devices, methods and compositions for reproductive organs PGF, GNRHR, PROX1 ESR1 216/4885KDM4E 3274/4885KMT2A 4546/4885
US-12533364-B2 Methods and compositions for testosterone production SHBG, FSHR, GNRHR ESR1 27/4885KDM4E 2825/4885KMT2A 3389/4885
US-20020137749-A1 Formulation for menopausal women SHBG, FABP6, BRCA1 ESR1 17/4885KDM4E 3618/4885KMT2A 3096/4885
US-20020173510-A1 Formulation for menopausal women SHBG, FABP6, BRCA1 ESR1 17/4885KDM4E 3618/4885KMT2A 3096/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.