SCHEMBL22066232

SCHEMBL22066232

CC(=O)Nc1ccc(S(=O)(=O)Nc2ccc(N)c(C)c2)cc1

nearest known ligand 0.77

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PKM P14618 2/20 0.77
ALDH1A1 P00352 3/20 0.63
LMNA P02545 3/20 0.60
SMN1; SMN2 Q16637 3/20 0.60
MAPK1 P28482 2/20 0.60
ALOX15 P16050 1/20 0.60
HTT P42858 1/20 0.60
MEN1 O00255 4/20 0.59
KMT2A Q03164 4/20 0.59
KDM4E B2RXH2 2/20 0.59
CYP3A4 P08684 1/20 0.59
HPGD P15428 1/20 0.59
TDP1 Q9NUW8 1/20 0.59
IDO1 P14902 1/20 0.57
RAB9A P51151 1/20 0.57
GAA P10253 1/20 0.57
GFER P55789 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28790906 0.84 FFAR4 (0.68) PKMALDH1A1LMNASMN1; SMN2MAPK1
SCHEMBL8921186 0.83 PKM (0.64) PKMALDH1A1LMNASMN1; SMN2MAPK1
SCHEMBL1832506 0.82 ALDH1A1 (0.57) PKMALDH1A1SMN1; SMN2ALOX15HTT
SCHEMBL7834756 0.81 LMNA (0.66) PKMALDH1A1LMNASMN1; SMN2MAPK1
SCHEMBL29118884 0.81 PKM (0.73) PKMALDH1A1LMNASMN1; SMN2MAPK1
SCHEMBL10572974 0.81 FFAR4 (0.68) PKMALDH1A1LMNASMN1; SMN2ALOX15
SCHEMBL7574036 0.80 PKM (0.68) PKMALDH1A1LMNASMN1; SMN2MAPK1
SCHEMBL14573241 0.80 PKM (0.56) PKMALDH1A1LMNASMN1; SMN2MAPK1
SCHEMBL4966207 0.80 KDM4E (0.69) PKMALDH1A1LMNASMN1; SMN2MAPK1
SCHEMBL9365750 0.79 PKM (0.73) PKMALDH1A1LMNASMN1; SMN2MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3663293-A1 SUBSTITUTED PENTA- AND HEXA-HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, DRUG COMBINATION AND USE THEREOF Xiamen University (CN) 2020-06-10 EP disclosed