SCHEMBL22069604

SCHEMBL22069604

CNCC(=O)Nc1ccc(Oc2ccc(Br)cc2)c(F)c1

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.51
MAPT P10636 3/20 0.51
MEN1 O00255 3/20 0.51
KMT2A Q03164 3/20 0.51
RAF1 P04049 2/20 0.49
MAPK3 P27361 1/20 0.49
FFAR1 O14842 5/20 0.48
PNLIP P16233 1/20 0.46
MET P08581 3/20 0.46
SLC1A3 P43003 1/20 0.44
SLC1A2 P43004 1/20 0.44
SLC1A1 P43005 1/20 0.44
GAA P10253 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
HPGD P15428 1/20 0.42
RAB9A P51151 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22069632 0.88 PNLIP (0.51) ALDH1A1MAPTFFAR1PNLIPMET
SCHEMBL22114313 0.88 MAPT (0.50) ALDH1A1MAPTMEN1KMT2ARAF1
SCHEMBL22114364 0.86 ALDH1A1 (0.48) ALDH1A1MAPTMEN1KMT2AHPGD
SCHEMBL22069654 0.86 FFAR1 (0.52) ALDH1A1MEN1KMT2AFFAR1PNLIP
SCHEMBL22069709 0.85 PNLIP (0.51) MAPTMEN1KMT2APNLIP
SCHEMBL22069696 0.85 RNF4 (0.51) ALDH1A1MAPTMEN1KMT2ARAF1
SCHEMBL22069658 0.84 FFAR1 (0.55) ALDH1A1MAPTMEN1KMT2ARAF1
SCHEMBL22069738 0.83 HTR2A (0.49) ALDH1A1FFAR1MET
SCHEMBL22069685 0.83 MET (0.46) MAPTMEN1KMT2AFFAR1PNLIP
SCHEMBL22069731 0.80 P2RX4 (0.54) FFAR1MET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3666769-A1 NOVEL CASPASE INHIBITORS RIJKSUNIVERSITEIT GRONINGEN (NL) 2020-06-17 EP disclosed
EP-3666769-A1 NOVEL CASPASE INHIBITORS RIJKSUNIVERSITEIT GRONINGEN (NL) 2020-06-17 EP disclosed