SCHEMBL22069738

SCHEMBL22069738

CNCC(=O)Nc1ccc(Oc2ccc(Cl)c(Cl)c2)c(F)c1

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 11/20 0.49
SLC6A4 P31645 11/20 0.49
KCNH2 Q12809 10/20 0.49
MET P08581 1/20 0.47
SCN9A Q15858 1/20 0.47
FFAR1 O14842 1/20 0.47
PARG Q86W56 1/20 0.46
CYP3A4 P08684 1/20 0.46
GRIN1 Q05586 1/20 0.43
GRIN2B Q13224 1/20 0.43
ALDH1A1 P00352 1/20 0.43
TSHR P16473 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22069632 0.88 PNLIP (0.51) HTR2ASLC6A4KCNH2METFFAR1
SCHEMBL22069652 0.87 MET (0.49) HTR2ASLC6A4KCNH2METSCN9A
SCHEMBL22069685 0.86 MET (0.46) METFFAR1PARGTSHR
SCHEMBL22069731 0.85 P2RX4 (0.54) METFFAR1PARG
SCHEMBL22069654 0.84 FFAR1 (0.52) METFFAR1PARGALDH1A1
SCHEMBL22069604 0.83 ALDH1A1 (0.51) METFFAR1ALDH1A1
SCHEMBL22069624 0.82 MAPT (0.49) FFAR1ALDH1A1TSHR
SCHEMBL22069658 0.82 FFAR1 (0.55) METFFAR1ALDH1A1TSHR
SCHEMBL22069626 0.81 MAPT (0.47) METFFAR1ALDH1A1TSHR
SCHEMBL22069653 0.80 L3MBTL1 (0.50) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3666769-A1 NOVEL CASPASE INHIBITORS RIJKSUNIVERSITEIT GRONINGEN (NL) 2020-06-17 EP disclosed
EP-3666769-A1 NOVEL CASPASE INHIBITORS RIJKSUNIVERSITEIT GRONINGEN (NL) 2020-06-17 EP disclosed