SCHEMBL22069731

SCHEMBL22069731

CNCC(=O)Nc1ccc(Oc2cccc(Cl)c2)c(F)c1

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
P2RX4 Q99571 13/20 0.54
CYP2C8 P10632 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2C9 P11712 1/20 0.50
ADRA2B P18089 1/20 0.50
HTR2C P28335 1/20 0.50
P2RX3 P56373 1/20 0.50
SLC6A3 Q01959 1/20 0.50
TMEM97 Q5BJF2 1/20 0.50
P2RX7 Q99572 1/20 0.50
FFAR1 O14842 4/20 0.48
MET P08581 1/20 0.46
PARG Q86W56 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22069685 0.90 MET (0.46) P2RX4FFAR1METPARG
SCHEMBL22069659 0.88 P2RX4 (0.54) P2RX4CYP2C8CYP2D6CYP2C9ADRA2B
SCHEMBL22069611 0.87 P2RX4 (0.57) P2RX4CYP2C8CYP2D6CYP2C9ADRA2B
SCHEMBL22069632 0.87 PNLIP (0.51) FFAR1METPARG
SCHEMBL22069738 0.85 HTR2A (0.49) FFAR1METPARG
SCHEMBL22069624 0.84 MAPT (0.49) FFAR1
SCHEMBL22069626 0.82 MAPT (0.47) FFAR1MET
SCHEMBL22069658 0.81 FFAR1 (0.55) FFAR1MET
SCHEMBL22069654 0.81 FFAR1 (0.52) FFAR1METPARG
SCHEMBL22069604 0.80 ALDH1A1 (0.51) FFAR1MET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3666769-A1 NOVEL CASPASE INHIBITORS RIJKSUNIVERSITEIT GRONINGEN (NL) 2020-06-17 EP disclosed
EP-3666769-A1 NOVEL CASPASE INHIBITORS RIJKSUNIVERSITEIT GRONINGEN (NL) 2020-06-17 EP disclosed