SCHEMBL22069652

SCHEMBL22069652

O=C(CCl)Nc1ccc(Oc2ccc(Cl)c(Cl)c2)c(F)c1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MET P08581 2/20 0.49
PARG Q86W56 1/20 0.48
MITF O75030 1/20 0.47
ALDH1A1 P00352 1/20 0.47
POLB P06746 1/20 0.47
MAPK1 P28482 1/20 0.47
HTT P42858 1/20 0.47
RNF4 P78317 1/20 0.47
SCN9A Q15858 1/20 0.46
CYP3A4 P08684 1/20 0.46
FNTA P49354 1/20 0.45
FNTB P49356 1/20 0.45
SLC2A1 P11166 1/20 0.45
PNLIP P16233 2/20 0.45
GSTO1 P78417 2/20 0.44
FFAR1 O14842 1/20 0.44
HTR2A P28223 3/20 0.44
SLC6A4 P31645 3/20 0.44
KCNH2 Q12809 3/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22069580 0.87 PNLIP (0.54) METPARGMITFALDH1A1POLB
SCHEMBL22069738 0.87 HTR2A (0.49) METPARGALDH1A1SCN9ACYP3A4
SCHEMBL22069703 0.85 MET (0.48) METPARGMITFALDH1A1POLB
SCHEMBL22069611 0.84 P2RX4 (0.57) METPARGMITFALDH1A1POLB
SCHEMBL22069696 0.84 RNF4 (0.51) METPARGMITFALDH1A1POLB
SCHEMBL22069558 0.83 FFAR1 (0.50) METPARGMITFALDH1A1POLB
SCHEMBL22069737 0.81 FFAR1 (0.53) METMITFALDH1A1POLBMAPK1
SCHEMBL22069574 0.81 ALDH1A1 (0.48) METPARGMITFALDH1A1POLB
SCHEMBL22114135 0.81 P2RX4 (0.52) METMITFALDH1A1POLBMAPK1
SCHEMBL4003878 0.78 CYP3A4 (0.71) ALDH1A1HTTCYP3A4GSTO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3666769-A1 NOVEL CASPASE INHIBITORS RIJKSUNIVERSITEIT GRONINGEN (NL) 2020-06-17 EP disclosed
EP-3666769-A1 NOVEL CASPASE INHIBITORS RIJKSUNIVERSITEIT GRONINGEN (NL) 2020-06-17 EP disclosed